SCHEMBL8634463

SCHEMBL8634463

COc1cc([N+](=O)[O-])ccc1C(=O)N1c2ccc(Cl)cc2CCCC1OCCCOS(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.35
MAPT P10636 3/20 0.35
MEN1 O00255 3/20 0.35
KCNMA1 Q12791 1/20 0.35
POLB P06746 2/20 0.34
TP53 P04637 3/20 0.34
ALDH1A1 P00352 5/20 0.34
NPC1 O15118 1/20 0.34
PYGL P06737 1/20 0.34
CYP3A4 P08684 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8627538 0.96 KCNMA1 (0.36) KMT2AMAPTMEN1KCNMA1POLB
SCHEMBL8627677 0.92 AVPR2 (0.38) KMT2AMAPTMEN1POLBTP53
SCHEMBL8634053 0.89 AVPR2 (0.41) KMT2AMAPTPOLBTP53
SCHEMBL8629507 0.88 KCNMA1 (0.36) KMT2AMAPTMEN1KCNMA1POLB
SCHEMBL8627401 0.88 AVPR2 (0.39) KMT2AMAPTMEN1TP53ALDH1A1
SCHEMBL8634460 0.87 MAPT (0.36) KMT2AMAPTMEN1KCNMA1POLB
SCHEMBL8627536 0.85 KCNMA1 (0.35) KMT2AMAPTMEN1KCNMA1POLB
SCHEMBL8627190 0.85 AVPR2 (0.42) KMT2AMAPTPOLBTP53
SCHEMBL8630395 0.84 PDK1 (0.35) KMT2AMAPTMEN1TP53ALDH1A1
SCHEMBL8629474 0.83 AVPR2 (0.51) MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed