SCHEMBL8634783

SCHEMBL8634783

C=CCOCC=C.Oc1ccccc1N1CCN(c2ccncc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.47
HTT P42858 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.41
DRD4 P21917 1/20 0.40
GFER P55789 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
METAP1 P53582 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CHKA P35790 1/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
HRH2 P25021 1/20 0.37
HRH1 P35367 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8636540 0.85 GAA (0.62) GAAHTTSMN1; SMN2DRD4GFER
SCHEMBL7399577 0.82 CHKA (0.43) GAASMN1; SMN2DRD4GFERMEN1
SCHEMBL8634780 0.79 SMN1; SMN2 (0.48) SMN1; SMN2DRD4METAP1MEN1KMT2A
Phenol SCHEMBL8634778 0.74 HRH3 (0.42) GAASMN1; SMN2DRD4METAP1MEN1
SCHEMBL8699660 0.73 GAA (0.37) GAAHTTDRD4GFERNPC1
SCHEMBL7329611 0.71 METAP1 (0.52) METAP1CHKAHRH2HRH1HRH3
Catechol SCHEMBL6545013 0.70 MAPT (0.48) GAAHTTSMN1; SMN2NPC1RAB9A
SCHEMBL11120307 0.70 GAA (0.70) GAAHTTSMN1; SMN2DRD4GFER
SCHEMBL4019882 0.70 GAA (0.70) GAAHTTSMN1; SMN2DRD4GFER
SCHEMBL17831308 0.67 CHKA (0.48) GAAHTTSMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed