SCHEMBL8635406

SCHEMBL8635406

COc1ccc(Cl)c(Oc2c(N)nc(N3CCOCC3)nc2COCC(O)CO)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 1/20 0.44
MAPT P10636 3/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PIK3CD O00329 6/20 0.36
PIK3CA P42336 6/20 0.36
PIK3CB P42338 4/20 0.36
HTR7 P34969 2/20 0.36
MAPK1 P28482 1/20 0.36
PIK3R1 P27986 1/20 0.36
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7850743 0.89 EDNRA (0.45) EDNRAMAPTL3MBTL1PIK3CDPIK3CA
SCHEMBL7849615 0.88 EDNRA (0.51) EDNRAMAPTL3MBTL1PIK3CDPIK3CA
SCHEMBL7853910 0.87 EDNRA (0.50) EDNRAMAPTL3MBTL1PIK3CDPIK3CA
SCHEMBL7849633 0.84 MAPT (0.47) EDNRAMAPTL3MBTL1PIK3CDPIK3CA
SCHEMBL7006902 0.81 EDNRA (0.70) EDNRAALDH1A1MEN1KMT2A
SCHEMBL7008278 0.81 EDNRA (0.70) EDNRAALDH1A1MEN1KMT2A
SCHEMBL7006905 0.81 EDNRA (0.70) EDNRAALDH1A1MEN1KMT2A
SCHEMBL7006907 0.80 EDNRA (0.42) EDNRAMAPTL3MBTL1PIK3CAHTR7
SCHEMBL7850538 0.79 MAPT (0.48) EDNRAMAPTL3MBTL1PIK3CDPIK3CA
SCHEMBL7849612 0.78 EDNRA (0.51) EDNRAMAPTL3MBTL1PIK3CDPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5837708-A CARDIOVASCULAR DISORDERS OF HYPERTENSION, ISCHEMIA, ANGINA PECTORIS AND VASOSPASMS HOFFMANN-LA ROCHE INC. (US) 1998-11-17 US disclosed