SCHEMBL7006907

SCHEMBL7006907

COc1ccc(Cl)c(Oc2c(COCC(O)CO)nc(N3CCOCC3)nc2N(CC(C)C)S(=O)(=O)c2ccccc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 2/20 0.42
PIK3CA P42336 2/20 0.35
MTOR P42345 1/20 0.35
RORC P51449 1/20 0.34
MAPT P10636 4/20 0.34
KMT2A Q03164 2/20 0.34
HTR7 P34969 2/20 0.34
GAA P10253 2/20 0.33
LMNA P02545 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
TNF P01375 1/20 0.33
NOD2 Q9HC29 1/20 0.33
NOD1 Q9Y239 1/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
OPRK1 P41145 1/20 0.33
EDNRB P24530 1/20 0.33
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7018075 0.92 EDNRA (0.48) EDNRAPIK3CAMTORRORCMAPT
SCHEMBL7012433 0.91 EDNRA (0.47) EDNRAPIK3CAMTORRORCMAPT
SCHEMBL7013473 0.88 EDNRA (0.44) EDNRAPIK3CAMTORRORCMAPT
SCHEMBL7013707 0.85 EDNRA (0.45) EDNRAPIK3CAMTORRORCMAPT
SCHEMBL7009897 0.83 EDNRA (0.43) EDNRAPIK3CAMTORRORCMAPT
SCHEMBL7008566 0.83 GAA (0.37) EDNRAMAPTKMT2AGAALMNA
SCHEMBL8635406 0.80 EDNRA (0.44) EDNRAPIK3CAMAPTKMT2AHTR7
SCHEMBL7850743 0.79 EDNRA (0.45) EDNRAPIK3CAMAPTKMT2AHTR7
SCHEMBL7006902 0.76 EDNRA (0.70) EDNRAKMT2ALMNAALDH1A1EDNRB
SCHEMBL7008278 0.76 EDNRA (0.70) EDNRAKMT2ALMNAALDH1A1EDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0601386-B1 Sulphonamides HOFFMANN LA ROCHE (CH) 2003-02-05 EP claimed
EP-0601386-A1 Sulphonamides F. HOFFMANN-LA ROCHE AG (CH) 1994-06-15 EP claimed
EP-0601386-B1 Sulphonamides HOFFMANN LA ROCHE (CH) 2003-02-05 EP disclosed
EP-0601386-A1 Sulphonamides F. HOFFMANN-LA ROCHE AG (CH) 1994-06-15 EP disclosed