SCHEMBL8635946

SCHEMBL8635946

NS(=O)(=O)c1ccccc1-n1nc(C(F)(F)F)cc1-c1cc(F)c(F)c(F)c1

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.53
PTGS1 P23219 6/20 0.53
PDPK1 O15530 4/20 0.51
CYP2C9 P11712 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8643945 0.89 PTGS2 (0.56) PTGS2PTGS1PDPK1CYP2C9
SCHEMBL8640374 0.88 PTGS2 (0.50) PTGS2PTGS1PDPK1
SCHEMBL8689089 0.88 PTGS2 (0.56) PTGS2PTGS1PDPK1
SCHEMBL8640768 0.88 PTGS2 (0.67) PTGS2PTGS1PDPK1CYP2C9
SCHEMBL5694290 0.87 PTGS2 (0.65) PTGS2PTGS1PDPK1CYP2C9
SCHEMBL8637251 0.86 PTGS2 (0.54) PTGS2PTGS1PDPK1
SCHEMBL8638758 0.86 PTGS2 (0.48) PTGS2PTGS1PDPK1
SCHEMBL8639187 0.86 PTGS2 (0.66) PTGS2PTGS1PDPK1CYP2C9
SCHEMBL8637765 0.86 PDPK1 (0.50) PTGS2PTGS1PDPK1
SCHEMBL8637585 0.86 PDPK1 (0.69) PTGS2PTGS1PDPK1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed