SCHEMBL8640374

SCHEMBL8640374

NS(=O)(=O)c1ccccc1-n1nc(C(F)(F)F)cc1-c1c(F)c(F)cc(F)c1F

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.50
PTGS1 P23219 7/20 0.50
PDPK1 O15530 4/20 0.48
F10 P00742 2/20 0.44
F2 P00734 1/20 0.44
KLKB1 P03952 1/20 0.44
PROC P04070 1/20 0.44
PRSS1 P07477 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8638758 0.93 PTGS2 (0.48) PTGS2PTGS1PDPK1F10F2
SCHEMBL8637765 0.93 PDPK1 (0.50) PTGS2PTGS1PDPK1
SCHEMBL8639142 0.92 PTGS2 (0.49) PTGS2PTGS1PDPK1F10
SCHEMBL8640038 0.89 PTGS2 (0.54) PTGS2PTGS1PDPK1
SCHEMBL8635946 0.88 PTGS2 (0.53) PTGS2PTGS1PDPK1
SCHEMBL8637343 0.88 PTGS2 (0.50) PTGS2PTGS1PDPK1F10
SCHEMBL8637251 0.86 PTGS2 (0.54) PTGS2PTGS1PDPK1F10F2
SCHEMBL8641753 0.86 PTGS2 (0.56) PTGS2PTGS1PDPK1F10F2
SCHEMBL8639323 0.86 PTGS2 (0.51) PTGS2PTGS1PDPK1
SCHEMBL8644146 0.85 PTGS2 (0.69) PTGS2PTGS1PDPK1F10F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed