SCHEMBL8637099

SCHEMBL8637099

Nc1ccc2nc(CCOc3ccc(Cc4ccccc4)cc3)[nH]c2c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 4/20 0.67
GRIN2B Q13224 4/20 0.67
MAPT P10636 8/20 0.65
PKM P14618 4/20 0.65
RAB9A P51151 4/20 0.65
SMN1; SMN2 Q16637 3/20 0.65
KDM4E B2RXH2 2/20 0.65
TDP1 Q9NUW8 2/20 0.65
ALDH1A1 P00352 2/20 0.65
GAA P10253 2/20 0.65
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
RAD52 P43351 2/20 0.52
UBE2N P61088 1/20 0.52
LMNA P02545 2/20 0.52
NPC1 O15118 2/20 0.52
HTT P42858 1/20 0.49
CYP1A2 P05177 1/20 0.48
POLB P06746 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8639346 0.91 GRIN1 (0.55) GRIN1GRIN2BMAPTPKMRAB9A
SCHEMBL8641196 0.85 GRIN1 (0.63) GRIN1GRIN2BMAPTRAB9ASMN1; SMN2
SCHEMBL8557293 0.81 MAPT (0.97) GRIN1GRIN2BMAPTPKMRAB9A
SCHEMBL7453184 0.81 GRIN1 (1.00) GRIN1GRIN2BMAPTPKMRAB9A
SCHEMBL6368842 0.77 MAPT (0.84) GRIN1GRIN2BMAPTPKMRAB9A
SCHEMBL8641842 0.75 LTA4H (0.51) MAPTRAB9AL3MBTL1LMNANPC1
SCHEMBL8640793 0.75 NPC1 (0.65) GRIN1GRIN2BMAPTRAB9ASMN1; SMN2
SCHEMBL27918353 0.75 GRIN1 (0.73) GRIN1GRIN2BMAPTPKMRAB9A
SCHEMBL8948422 0.74 NPC1 (0.71) GRIN1GRIN2BMAPTRAB9ASMN1; SMN2
SCHEMBL8641659 0.72 GRIN1 (0.66) GRIN1GRIN2BMAPTRAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5723492-A LTA4 hydrolase inhibitor pharmaceutical compositions and methods of use G.D. SEARLE & CO. (US) 1998-03-03 US disclosed
US-5719306-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed