SCHEMBL8637656

SCHEMBL8637656

CNS(=O)(=O)c1ccc(-c2cc(C(F)(F)F)nn2NS(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 11/20 0.48
PDPK1 O15530 5/20 0.46
PTGS1 P23219 7/20 0.46
KIF11 P52732 1/20 0.45
CYP2C9 P11712 2/20 0.42
ALOX5 P09917 2/20 0.41
PTGES O14684 1/20 0.41
HDAC3 O15379 1/20 0.41
CA12 O43570 1/20 0.41
PDE5A O76074 1/20 0.41
ABCB11 O95342 1/20 0.41
MT-CO2 P00403 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
LMNA P02545 1/20 0.41
CA3 P07451 1/20 0.41
CYP3A4 P08684 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
CYP2D6 P10635 1/20 0.41
ADRB3 P13945 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8640765 0.90 PTGS1 (0.51) PTGS2PDPK1PTGS1RXRANR1H2
SCHEMBL8652506 0.89 PTGS2 (0.54) PTGS2PDPK1PTGS1RXRANR1H2
SCHEMBL7135445 0.89 PTGS2 (0.51) PTGS2PDPK1PTGS1CYP2C9ALOX5
SCHEMBL8636828 0.88 PDPK1 (0.61) PTGS2PDPK1PTGS1CYP2C9ALOX5
SCHEMBL8351386 0.88 PTGS2 (0.49) PTGS2PDPK1PTGS1RXRANR1H2
SCHEMBL8641577 0.88 PTGS2 (0.49) PTGS2PDPK1PTGS1CYP2C9RXRA
SCHEMBL8638028 0.87 PDPK1 (0.52) PTGS2PDPK1PTGS1CYP2C9RXRA
SCHEMBL8640576 0.87 PTGS2 (0.55) PTGS2PDPK1PTGS1CA12CA2
SCHEMBL8638817 0.87 PTGS2 (0.46) PTGS2PDPK1PTGS1ALOX5RXRA
SCHEMBL8639795 0.87 PTGS2 (0.50) PTGS2PDPK1PTGS1CYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed