SCHEMBL8637722

SCHEMBL8637722

O=S(=O)(Nn1nc(CCCO)cc1-c1ccccc1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.46
CA2 P00918 5/20 0.46
CA9 Q16790 4/20 0.46
ALOX5 P09917 1/20 0.43
PTGS2 P35354 7/20 0.40
EPHX2 P34913 7/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
MALT1 Q9UDY8 1/20 0.37
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36
MMP13 P45452 1/20 0.36
AKR1C3 P42330 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8639925 0.92 CA1 (0.40) CA1CA2CA9ALOX5PTGS2
SCHEMBL8689039 0.87 CA1 (0.53) CA1CA2CA9PTGS2MALT1
SCHEMBL8693706 0.84 ALDH1A1 (0.36) CA1CA2CA9ALOX5PTGS2
SCHEMBL8688890 0.82 CA1 (0.42) CA1CA2CA9ALOX5PTGS2
SCHEMBL8688829 0.82 PTGS2 (0.52) CA1CA2CA9ALOX5PTGS2
SCHEMBL8689453 0.80 EPHX2 (0.40) CA1CA2CA9ALOX5PTGS2
SCHEMBL7924388 0.80 PTGS2 (0.51) CA1CA2CA9ALOX5PTGS2
SCHEMBL6531309 0.80 CA1 (0.51) CA1CA2CA9PTGS2MALT1
SCHEMBL8692354 0.79 EPHX2 (0.41) CA1CA2CA9PTGS2EPHX2
SCHEMBL8693633 0.79 NMT1 (0.39) CA1CA2CA9ALOX5PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed