SCHEMBL8637994

SCHEMBL8637994

CCOP(=O)(OCC)N(CC)CCCN(C/C=C/CN(CCCN(CC)P(=O)(OCC)OCC)P(=O)(OCC)OCC)P(=O)(OCC)OCC

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.32
TP53 P04637 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8641792 0.86 TDP1 (0.39) TSHRTDP1
SCHEMBL8641789 0.86 TDP1 (0.39) TSHRTDP1
SCHEMBL21049917 0.81 TSHR (0.37) TSHRTP53TDP1
SCHEMBL8641772 0.80 TDP1 (0.43) TDP1
SCHEMBL8641794 0.80 TDP1 (0.43) TDP1
SCHEMBL3289373 0.76 TSHR (0.48) TSHRTP53TDP1
SCHEMBL6988924 0.69 TSHR (0.37) TSHRTP53TDP1
SCHEMBL12207660 0.68 TSHR (0.43) TSHRTP53TDP1
SCHEMBL3103434 0.66 ACHE (0.40) TSHRTP53TDP1
SCHEMBL6985563 0.65 TSHR (0.40) TSHRTP53TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686143-B1 UNSATURATE AMINO COMPOUNDS FOR USE AS ANTICANCER AND ANTIPROTOZOIC AGENT CIBA GEIGY AG (CH) 1998-08-12 EP disclosed
US-5627215-A Unsaturate amino compounds for use as anticancer and antiprotozoic agent CIBA-GEIGY CORPORATION (US) 1997-05-06 US disclosed
EP-0686143-A1 UNSATURATE AMINO COMPOUNDS FOR USE AS ANTICANCER AND ANTIPROTOZOIC AGENT Novartis AG (CH) 1995-12-13 EP disclosed
WO-1995018091-A1 UNSATURATE AMINO COMPOUNDS FOR USE AS ANTICANCER AND ANTIPROTOZOIC AGENT CIBA-GEIGY AG (CH) 1995-07-06 WO disclosed