SCHEMBL6988924

SCHEMBL6988924

CCOP(=O)(OCC)N(CCCN)CCCN

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.37
CYP1A2 P05177 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TP53 P04637 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
GABBR2 O75899 3/20 0.33
GABBR1 Q9UBS5 3/20 0.33
GABRR1 P24046 1/20 0.32
ACHE P22303 1/20 0.31
THPO P40225 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985563 0.87 TSHR (0.40) TSHRMEN1KMT2ATP53TDP1
SCHEMBL24268058 0.78 GABBR2 (0.33) TSHRCYP1A2GABBR2GABBR1GABRR1
SCHEMBL12207660 0.78 TSHR (0.43) TSHRMEN1KMT2ATP53TDP1
SCHEMBL21049917 0.75 TSHR (0.37) TSHRMEN1KMT2ATP53TDP1
SCHEMBL3103434 0.75 ACHE (0.40) TSHRMEN1KMT2ATP53TDP1
SCHEMBL6990161 0.74 PPARD (0.46) TSHRMEN1KMT2ATP53TDP1
SCHEMBL3289373 0.72 TSHR (0.48) TSHRMEN1KMT2ATP53TDP1
SCHEMBL8637994 0.69 TSHR (0.32) TSHRTP53TDP1
SCHEMBL6990204 0.69 ACHE (0.42) TSHRMEN1KMT2ATP53TDP1
SCHEMBL11154240 0.69 PPARD (0.44) TSHRTP53TDP1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0739345-B1 CYCLIC POLYAMINES ANORMED INC (CA) 2003-04-09 EP disclosed
US-5698546-A Cyclic polyamines JOHNSON MATTHEY PUBLIC LIMTED COMPANY (GB) 1997-12-16 US disclosed
EP-0739345-A1 CYCLIC POLYAMINES JOHNSON MATTHEY PUBLIC LIMITED COMPANY (GB) 1996-10-30 EP disclosed
WO-1995018808-A1 CYCLIC POLYAMINES JOHNSON MATTHEY PUBLIC LIMITED COMPANY (GB) 1995-07-13 WO disclosed