SCHEMBL8638423

SCHEMBL8638423

O=C(NCCOc1ccc(Oc2ccccc2)cc1)C1CCCNC1

nearest known ligand 0.66

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.66
RAB9A P51151 4/20 0.66
SMN1; SMN2 Q16637 3/20 0.66
PKM P14618 1/20 0.66
EPHX2 P34913 1/20 0.66
KMT2A Q03164 4/20 0.54
MEN1 O00255 2/20 0.54
F10 P00742 1/20 0.48
ALOX15 P16050 1/20 0.46
MTNR1A P48039 1/20 0.45
MTNR1B P49286 1/20 0.45
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
REN P00797 1/20 0.43
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8639341 0.97 NPC1 (0.61) NPC1RAB9ASMN1; SMN2PKMEPHX2
SCHEMBL8641245 0.89 NPC1 (0.60) NPC1RAB9ASMN1; SMN2PKMEPHX2
SCHEMBL8640087 0.86 SMN1; SMN2 (0.68) NPC1RAB9ASMN1; SMN2PKMEPHX2
SCHEMBL8640783 0.86 SMN1; SMN2 (0.56) NPC1RAB9ASMN1; SMN2PKMEPHX2
SCHEMBL9730574 0.84 NPC1 (0.77) NPC1RAB9ASMN1; SMN2PKMEPHX2
SCHEMBL8641864 0.82 SMN1; SMN2 (0.63) NPC1RAB9ASMN1; SMN2PKMEPHX2
SCHEMBL8641254 0.82 SMN1; SMN2 (0.56) NPC1RAB9ASMN1; SMN2PKMEPHX2
SCHEMBL17842262 0.80 RAB9A (0.75) NPC1RAB9ASMN1; SMN2PKMEPHX2
SCHEMBL22447941 0.80 NPC1 (1.00) NPC1RAB9ASMN1; SMN2PKMEPHX2
SCHEMBL23975373 0.78 SMN1; SMN2 (0.89) NPC1RAB9ASMN1; SMN2PKMEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5723492-A LTA4 hydrolase inhibitor pharmaceutical compositions and methods of use G.D. SEARLE & CO. (US) 1998-03-03 US disclosed
US-5719306-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed
EP-0804427-A1 LTA4 HYDROLASE INHIBITORS G.D. SEARLE & CO. (US) 1997-11-05 EP disclosed
WO-1996011192-A1 LTA4 HYDROLASE INHIBITORS G.D. SEARLE & CO. (US) 1996-04-18 WO disclosed