SCHEMBL8639153

SCHEMBL8639153

COc1cc(Cl)ccc1-c1cc(C(F)(F)F)nn1NS(=O)(=O)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.45
PTGS1 P23219 3/20 0.39
ATM Q13315 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
IGF1R P08069 1/20 0.39
AVPR2 P30518 1/20 0.38
GPR27 Q9NS67 1/20 0.38
MAPT P10636 3/20 0.38
POLB P06746 1/20 0.38
TSHR P16473 2/20 0.38
NPC1 O15118 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
THPO P40225 1/20 0.38
BLM P54132 1/20 0.38
PMP22 Q01453 1/20 0.38
HIF1A Q16665 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8690933 0.89 PTGS2 (0.45) PTGS2PTGS1L3MBTL1MAPTPOLB
SCHEMBL8639423 0.89 PTGS2 (0.48) PTGS2PTGS1MAPTPOLBNPSR1
SCHEMBL8636816 0.88 PTGS2 (0.56) PTGS2PTGS1L3MBTL1MAPTNPSR1
SCHEMBL8640002 0.86 PTGS2 (0.42) PTGS2PTGS1GPR27
SCHEMBL8635926 0.86 PTGS2 (0.53) PTGS2PTGS1POLBFLT1FLT4
SCHEMBL8637076 0.84 PTGS2 (0.43) PTGS2PTGS1FLT1FLT4KDR
SCHEMBL8641742 0.84 PTGS2 (0.40) PTGS2PTGS1AVPR2GPR27MAPT
SCHEMBL8689324 0.82 PTGS2 (0.45) PTGS2PTGS1MAPTPOLBTSHR
SCHEMBL8641086 0.81 PTGS2 (0.44) PTGS2PTGS1MAPTSCN9ASMN1; SMN2
SCHEMBL8639795 0.80 PTGS2 (0.50) PTGS2PTGS1TSHRCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed