SCHEMBL8640229

SCHEMBL8640229

CCCOC(=O)N[C@H]1CCn2c(cc3ccccc32)C1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.43
HTR2C P28335 2/20 0.43
KCNA3 P22001 1/20 0.39
MCHR1 Q99705 1/20 0.39
HSD11B1 P28845 1/20 0.39
SIGMAR1 Q99720 9/20 0.38
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSK P43235 1/20 0.38
EPHX1 P07099 1/20 0.38
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6590757 0.83 KCNA3 (0.50) KCNA3SIGMAR1CTSKCNR1CNR2
SCHEMBL3150583 0.74 KDM4E (0.47) KDM4E
SCHEMBL8656217 0.72 SIGMAR1 (0.42) HTR2AHTR2CSIGMAR1
SCHEMBL6015848 0.71 SIGMAR1 (0.44) HTR2AHTR2CSIGMAR1
SCHEMBL8319222 0.71 SIGMAR1 (0.44) HTR2AHTR2CSIGMAR1
SCHEMBL8653533 0.70 ALDH1A1 (0.48) KDM4E
SCHEMBL8653071 0.70 ACACB (0.50) KDM4E
SCHEMBL8452782 0.68 HTR2A (0.44) HTR2AHTR2CSIGMAR1
SCHEMBL8454162 0.68 HTR2A (0.44) HTR2AHTR2CSIGMAR1
SCHEMBL30684404 0.68 HTR2A (0.44) HTR2AHTR2CSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721230-A ANTIINFLAMMATORY AGENT, VIRICIDES; TREATING CARDIOVASCULAR DISORDER, RESPIRATORY SYSTEM DISORDER, THROMBOSIS, DIABETES, ALOPECIA HOFFMANN-LA ROCHE INC. (US) 1998-02-24 US disclosed