SCHEMBL8640518

SCHEMBL8640518

CSc1ccccc1-c1cc(C(F)(F)F)nn1NS(=O)(=O)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
PTGS2 P35354 12/20 0.39
PTGS1 P23219 7/20 0.39
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
PDPK1 O15530 1/20 0.35
FFAR4 Q5NUL3 1/20 0.34
RXRA P19793 1/20 0.34
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8639293 0.85 PTGS2 (0.54) PTGS2PTGS1PDPK1FFAR4
SCHEMBL8644144 0.83 PTGS2 (0.53) PTGS2PTGS1PDPK1FFAR4
SCHEMBL8688501 0.83 PTGS2 (0.44) ALDH1A1SMN1; SMN2PTGS2PTGS1KDM4E
SCHEMBL8688820 0.83 PTGS2 (0.56) ALDH1A1SMN1; SMN2PTGS2PTGS1KDM4E
SCHEMBL8689466 0.83 PTGS2 (0.46) ALDH1A1SMN1; SMN2PTGS2PTGS1KDM4E
SCHEMBL8641739 0.82 PTGS2 (0.54) PTGS2PTGS1PDPK1RXRANR1H2
SCHEMBL8691654 0.82 PTGS2 (0.45) ALDH1A1SMN1; SMN2PTGS2PTGS1KDM4E
SCHEMBL8636816 0.82 PTGS2 (0.56) ALDH1A1SMN1; SMN2PTGS2PTGS1KDM4E
SCHEMBL8641068 0.82 PTGS2 (0.53) ALDH1A1SMN1; SMN2PTGS2PTGS1KDM4E
SCHEMBL8641750 0.81 PTGS2 (0.42) ALDH1A1SMN1; SMN2PTGS2PTGS1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed