SCHEMBL8640692

SCHEMBL8640692

COc1c(C)cc(-c2cc(C(F)(F)F)nn2NS(=O)(=O)c2ccccc2)cc1C

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.48
PTGS1 P23219 7/20 0.45
MAPT P10636 2/20 0.39
THRB P10828 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PDPK1 O15530 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8688800 0.93 PTGS2 (0.58) PTGS2PTGS1MAPT
SCHEMBL8689085 0.89 PTGS2 (0.44) PTGS2PTGS1MAPTTHRBSMN1; SMN2
SCHEMBL8689331 0.88 PTGS2 (0.49) PTGS2PTGS1MAPT
SCHEMBL8639246 0.87 PTGS2 (0.56) PTGS2PTGS1MAPTTHRBSMN1; SMN2
SCHEMBL8641600 0.85 PTGS2 (0.44) PTGS2PTGS1SMN1; SMN2PDPK1
SCHEMBL27967579 0.85 PDPK1 (0.45) PTGS2PTGS1PDPK1
SCHEMBL7868758 0.84 PTGS2 (0.53) PTGS2PTGS1MAPTSMN1; SMN2
SCHEMBL8640765 0.84 PTGS1 (0.51) PTGS2PTGS1SMN1; SMN2PDPK1
SCHEMBL8636729 0.83 PTGS2 (0.43) PTGS2PTGS1PDPK1
SCHEMBL7135445 0.83 PTGS2 (0.51) PTGS2PTGS1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed