SCHEMBL8640694

SCHEMBL8640694

COc1c(C)cc(-c2cc(C(F)(F)F)nn2-c2ccccc2S(N)(=O)=O)cc1C

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.61
PTGS1 P23219 8/20 0.53
PDPK1 O15530 3/20 0.47
PTGES O14684 1/20 0.47
HDAC3 O15379 1/20 0.47
CA12 O43570 1/20 0.47
PDE5A O76074 1/20 0.47
ABCB11 O95342 1/20 0.47
MT-CO2 P00403 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
LMNA P02545 1/20 0.47
CA3 P07451 1/20 0.47
CYP3A4 P08684 1/20 0.47
ALOX5 P09917 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
ADRB3 P13945 1/20 0.47
ALOX15 P16050 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8688801 0.93 PTGS2 (0.72) PTGS2PTGS1
SCHEMBL8689089 0.90 PTGS2 (0.56) PTGS2PTGS1PDPK1
SCHEMBL8689333 0.89 PTGS2 (0.62) PTGS2PTGS1PDPK1
SCHEMBL8639247 0.88 PTGS2 (0.70) PTGS2PTGS1PDPK1PTGESHDAC3
SCHEMBL8641602 0.86 PTGS2 (0.53) PTGS2PTGS1PDPK1PTGESHDAC3
SCHEMBL8635878 0.85 PTGS2 (0.69) PTGS2PTGS1PDPK1CYP3A4CYP2C9
SCHEMBL8688454 0.84 PTGS2 (0.52) PTGS2PTGS1PDPK1PTGESHDAC3
SCHEMBL8636734 0.84 PTGS2 (0.52) PTGS2PTGS1PDPK1PTGESHDAC3
SCHEMBL29502699 0.84 PTGS2 (0.66) PTGS2PTGS1PDPK1PTGESHDAC3
SCHEMBL6912425 0.84 PTGS2 (0.66) PTGS2PTGS1PDPK1PTGESHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed