SCHEMBL8640873

SCHEMBL8640873

CCc1nc2nc(CO)cc(C)c2[nH]1

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 8/20 0.68
ADORA3 P0DMS8 7/20 0.47
ADORA2A P29274 6/20 0.47
NOS1 P29475 2/20 0.39
NOS2 P35228 2/20 0.39
NOS3 P29474 1/20 0.35
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33
DYRK1A Q13627 1/20 0.33
CDK1 P06493 1/20 0.32
CCNB1 P14635 1/20 0.32
CCNA2 P20248 1/20 0.32
CDK2 P24941 1/20 0.32
ADORA2B P29275 1/20 0.32
DDAH1 O94760 1/20 0.32
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30
HCAR2 Q8TDS4 1/20 0.30
TACR2 P21452 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8639237 0.84 ADORA1 (0.49) ADORA1ADORA3ADORA2ANOS1NOS2
SCHEMBL5091129 0.81 ADORA1 (1.00) ADORA1ADORA3ADORA2ANOS1NOS2
SCHEMBL3217333 0.78 ADORA1 (0.70) ADORA1ADORA3ADORA2ANOS1NOS2
SCHEMBL3210466 0.78 ADORA1 (0.70) ADORA1ADORA3ADORA2ANOS1NOS2
SCHEMBL7387472 0.76 ADORA1 (0.62) ADORA1ADORA3ADORA2ANOS1NOS2
Hydrochloric Acid SCHEMBL9597611 0.75 ADORA1 (0.60) ADORA1ADORA3ADORA2ANOS1NOS2
SCHEMBL7016763 0.74 ADORA1 (0.64) ADORA1ADORA3ADORA2ANOS1NOS2
SCHEMBL9597257 0.73 ADORA1 (0.57) ADORA1ADORA3ADORA2AGAAKMT2A
SCHEMBL7018191 0.73 ADORA1 (0.57) ADORA1ADORA3ADORA2ANOS1NOS2
SCHEMBL31569110 0.71 ADORA1 (0.47) ADORA1ADORA3ADORA2ANOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849753-A Pyridyl imidazole derivatives and processes for the preparation thereof KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1998-12-15 US disclosed
EP-0743943-A1 PYRIDYL IMIDAZOLE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1996-11-27 EP disclosed
WO-1995021838-A1 PYRIDYL IMIDAZOLE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1995-08-17 WO disclosed