SCHEMBL8639237

SCHEMBL8639237

CCCCc1nc2nc(CO)cc(C)c2[nH]1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 4/20 0.49
PI4KA P42356 1/20 0.43
PI4K2B Q8TCG2 1/20 0.43
PI4K2A Q9BTU6 1/20 0.43
PI4KB Q9UBF8 1/20 0.43
ADORA3 P0DMS8 3/20 0.41
ADORA2A P29274 3/20 0.41
NOS1 P29475 2/20 0.41
NOS2 P35228 2/20 0.41
GPR84 Q9NQS5 5/20 0.39
NOS3 P29474 1/20 0.37
ALDH1A1 P00352 1/20 0.36
MAPK1 P28482 1/20 0.36
GSK3B P49841 1/20 0.35
PARP1 P09874 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8640873 0.84 ADORA1 (0.68) ADORA1ADORA3ADORA2ANOS1NOS2
SCHEMBL8638332 0.83 ADORA1 (0.71) ADORA1PI4KAPI4K2BPI4K2API4KB
SCHEMBL5098257 0.73 ADORA1 (0.75) ADORA1PI4KAPI4K2BPI4K2API4KB
SCHEMBL8641790 0.73 PARP1 (0.39) PI4KAPI4K2BPI4K2API4KBNOS1
SCHEMBL9041424 0.73 NOS1 (0.56) ADORA1PI4KAPI4K2BPI4K2API4KB
SCHEMBL7386115 0.71 ADORA1 (0.53) ADORA1PI4KAPI4K2BPI4K2API4KB
SCHEMBL7383805 0.71 ADORA1 (0.53) ADORA1PI4KAPI4K2BPI4K2API4KB
SCHEMBL7383935 0.70 ADORA1 (0.48) ADORA1PI4KAPI4K2BPI4K2API4KB
SCHEMBL7852563 0.69 ADORA3 (0.48) ADORA1PI4KAPI4K2BPI4K2API4KB
SCHEMBL7851022 0.69 GCGR (0.48) ADORA1PI4KAPI4K2BPI4K2API4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849753-A Pyridyl imidazole derivatives and processes for the preparation thereof KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1998-12-15 US disclosed
EP-0743943-A1 PYRIDYL IMIDAZOLE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1996-11-27 EP disclosed
WO-1995021838-A1 PYRIDYL IMIDAZOLE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1995-08-17 WO disclosed