SCHEMBL864368

SCHEMBL864368

CNc1cc(Cl)c(C)cc1N

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD44 P16070 1/20 0.60
CYP3A4 P08684 3/20 0.40
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2A Q12879 1/20 0.36
GRIN2B Q13224 1/20 0.36
GRIN2C Q14957 1/20 0.36
GRIN3A Q8TCU5 1/20 0.36
PRKCI P41743 1/20 0.36
ALDH1A1 P00352 5/20 0.35
GAA P10253 2/20 0.35
KDM4E B2RXH2 2/20 0.33
LMNA P02545 2/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B2 P37059 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11816340 0.91 CD44 (0.60) CD44CYP3A4TSHRMAPK1GRIN2D
SCHEMBL31213265 0.84 GAA (0.46) CD44CYP3A4TSHRMAPK1PRKCI
SCHEMBL932424 0.84 GAA (0.46) CD44CYP3A4TSHRMAPK1PRKCI
Hydrochloric Acid SCHEMBL15158295 0.82 GAA (0.43) CD44CYP3A4TSHRMAPK1PRKCI
SCHEMBL6983173 0.81 TSHR (0.50) CD44CYP3A4TSHRMAPK1PRKCI
Hydrochloric Acid SCHEMBL11754022 0.79 TSHR (0.48) CD44CYP3A4TSHRMAPK1PRKCI
SCHEMBL12656572 0.79 CD44 (0.42) CD44CYP3A4MAPK1GRIN2DGRIN3B
Hydrochloric Acid SCHEMBL11754014 0.79 TSHR (0.48) CD44CYP3A4TSHRMAPK1PRKCI
SCHEMBL19199592 0.79 CD44 (0.42) CD44CYP3A4MAPK1GRIN2DGRIN3B
SCHEMBL13497800 0.78 CD44 (0.54) CD44CYP3A4TSHRMAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021130731-A1 SUBSTITUTED TRICYCLIC COMPOUNDS LUPIN LIMITED (IN) 2021-07-01 WO disclosed
EP-3763706-A1 PARASITICIDAL COMPOSITIONS COMPRISING BENZIMIDAZOLE DERIVATIVES, METHODS AND USES THEREOF Boehringer Ingelheim Animal Health USA Inc. (US) 2021-01-13 EP disclosed
EP-3453702-A2 PARASITICIDAL COMPOSITIONS COMPRISING BENZIMIDAZOLE DERIVATIVES, METHODS AND USES THEREOF Merial, Inc. (US) 2019-03-13 EP disclosed
US-20120077781-A1 FLAVIN DERIVATIVES GADWOOD ROBERT (US) 2012-03-29 US disclosed
US-20120077781-A1 FLAVIN DERIVATIVES GADWOOD ROBERT (US) 2012-03-29 US disclosed
US-20120077781-A1 FLAVIN DERIVATIVES GADWOOD ROBERT (US) 2012-03-29 US disclosed
WO-2010019208-A1 FLAVIN DERIVATIVES BIORELIX PHARMACEUTICALS, INC. (US) 2010-02-18 WO disclosed
US-3931215-A OPTICAL BRIGHTENERS HOECHST AKTIENGESELLSCHAFT (DT) 1976-01-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120077781-A1 FLAVIN DERIVATIVES BLVRB, FLAD1, FDPS CD44 3883/4885CYP3A4 415/4885TSHR 2380/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.