SCHEMBL8644251

SCHEMBL8644251

CCN1CCCC1(CO)Oc1ccc(Cc2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 13/20 0.42
HRH3 Q9Y5N1 2/20 0.38
KMT2A Q03164 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3134727 0.67 DRD2 (0.36) KDM4EALDH1A1CYP2D6
SCHEMBL6129775 0.66 OPRM1 (0.39)
SCHEMBL25051426 0.66 OPRM1 (0.39)
SCHEMBL14833411 0.64 DRD2 (0.38)
SCHEMBL3124211 0.63 OPRM1 (0.34) LTA4HKMT2AKDM4EMEN1ALDH1A1
SCHEMBL24998567 0.63 MEN1 (0.41) KMT2AMEN1ALDH1A1CYP2D6
SCHEMBL14058149 0.63 OPRL1 (0.34)
SCHEMBL25000121 0.62 CYP2D6 (0.43) KMT2AMEN1ALDH1A1CYP2D6
SCHEMBL31105377 0.62 CYP2D6 (0.43) KMT2AMEN1ALDH1A1CYP2D6
SCHEMBL12672699 0.62 MEN1 (0.45) KMT2AMEN1ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5723492-A LTA4 hydrolase inhibitor pharmaceutical compositions and methods of use G.D. SEARLE & CO. (US) 1998-03-03 US disclosed
US-5719306-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed