SCHEMBL8644292

SCHEMBL8644292

COc1ccc(CCC(=O)C(NC(=O)c2ccc(C(=N)N)cc2)(Oc2ccccc2)C(=O)O)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.47
ITGA2B P08514 3/20 0.47
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
SCN5A Q14524 1/20 0.45
SCN2A Q99250 1/20 0.45
GAA P10253 2/20 0.44
ALDH1A1 P00352 3/20 0.43
MAPT P10636 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
PRSS1 P07477 1/20 0.41
PRSS2 P07478 1/20 0.41
PRSS3 P35030 1/20 0.41
F2 P00734 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8646799 0.99 ITGB3 (0.46) ITGB3ITGA2BNPC1RAB9ASCN5A
SCHEMBL8646001 0.92 ITGB3 (0.45) ITGB3ITGA2BALDH1A1KDM4EF2
Hydrochloric Acid SCHEMBL8647767 0.91 ITGB3 (0.44) ITGB3ITGA2BALDH1A1KDM4EF2
SCHEMBL8644198 0.85 F10 (0.40) ITGB3ITGA2BPRSS1F2F10
SCHEMBL8644302 0.85 NPC1 (0.42) NPC1RAB9ASCN5ASCN2AGAA
Hydrochloric Acid SCHEMBL8646804 0.84 NPC1 (0.42) NPC1RAB9ASCN5ASCN2AGAA
Trifluoroacetic Acid SCHEMBL8644121 0.83 KLK1 (0.41) ITGB3ITGA2BF2F10
Trifluoroacetic Acid SCHEMBL8646468 0.83 KLK1 (0.43) ITGB3ITGA2BF2F10
SCHEMBL8645969 0.82 F10 (0.40) ITGB3ITGA2BPRSS1PRSS2PRSS3
Hydrochloric Acid SCHEMBL8644799 0.81 F10 (0.40) ITGB3ITGA2BPRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726185-A BINDING OF ADHESIVE PROTEINS TO BLOOD PLATELET AGGREGATION AND CELL TO CELL ADHESION HOFFMANN-LA ROCHE INC. (US) 1998-03-10 US disclosed