SCHEMBL8645744

SCHEMBL8645744

O=C(O)Cc1ccc2cccccc1-2

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.55
ABCC4 O15439 1/20 0.55
LMNA P02545 1/20 0.55
GAA P10253 1/20 0.55
TSHR P16473 1/20 0.55
HTT P42858 1/20 0.55
KMT2A Q03164 1/20 0.53
AKR1B1 P15121 2/20 0.52
PTGER1 P34995 2/20 0.51
PTGER4 P35408 2/20 0.51
PTGER3 P43115 2/20 0.51
PTGER2 P43116 2/20 0.51
MMP1 P03956 1/20 0.49
MMP2 P08253 1/20 0.49
MMP3 P08254 1/20 0.49
MMP9 P14780 1/20 0.49
MMP8 P22894 1/20 0.49
MMP12 P39900 1/20 0.49
MMP13 P45452 1/20 0.49
MMP14 P50281 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5961842 0.94 PTGS1 (0.59) PTGS1ABCC4LMNAGAATSHR
SCHEMBL538512 0.94 KMT2A (0.60) PTGS1ABCC4LMNAGAATSHR
Hydrochloric Acid SCHEMBL11895689 0.92 KMT2A (0.58) PTGS1ABCC4LMNAGAATSHR
SCHEMBL29512995 0.92 KMT2A (0.58) PTGS1ABCC4LMNAGAATSHR
SCHEMBL28594606 0.92 KMT2A (0.58) PTGS1ABCC4LMNAGAATSHR
SCHEMBL27701716 0.92 KMT2A (0.58) PTGS1ABCC4LMNAGAATSHR
Ammonia Solution, Strong SCHEMBL27926479 0.92 KMT2A (0.58) PTGS1ABCC4LMNAGAATSHR
Ethane SCHEMBL28588588 0.90 PTGS1 (0.57) PTGS1ABCC4LMNAGAATSHR
SCHEMBL28408449 0.86 PTGS1 (0.66) PTGS1ABCC4LMNAGAATSHR
SCHEMBL7601609 0.86 AKR1B1 (0.57) PTGS1ABCC4LMNAGAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1649875-A 2-thia-dibenzoazulenes as inhibitors of tumour necrosis factor production and intermediates for the preparation thereof PLIVA D D (HR) 2005-08-03 CN claimed
CN-101805283-B 1,4-dihydropyridines compound containing azulene structure and preparation method thereof UNIV SHANGHAI 2013-01-02 CN disclosed
CN-101805283-A 1,4-dihydropyridines compound containing azulene structure and preparation method thereof UNIV SHANGHAI 2010-08-18 CN disclosed
CN-1649875-A 2-thia-dibenzoazulenes as inhibitors of tumour necrosis factor production and intermediates for the preparation thereof PLIVA D D (HR) 2005-08-03 CN disclosed
CN-1345312-A Dibenzoazulene derivatives for treating thrombosis, osteoporosis arteriosclerosis MERCK PATENT GMBH (DE) 2002-04-17 CN disclosed
US-5843999-A 2-phenylazulene derivatives and a manufacturing method of these compounds KOTOBUKI SEIYAKU CO., LTD. (JP) 1998-12-01 US disclosed