SCHEMBL8648609

SCHEMBL8648609

COc1cc2ncnc(N3c4ccccc4[C@@H](C)[C@@H]3C)c2cc1OC

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.54
CSF1R P07333 1/20 0.53
ACHE P22303 6/20 0.51
BACE1 P56817 6/20 0.51
PDE10A Q9Y233 5/20 0.50
KIT P10721 1/20 0.49
ATM Q13315 2/20 0.48
RET P07949 1/20 0.47
KIF5B P33176 1/20 0.47
KDR P35968 1/20 0.47
HTR1A P08908 1/20 0.47
HTR7 P34969 1/20 0.47
PDE3A Q14432 1/20 0.47
AURKA O14965 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8649524 1.00 EGFR (0.54) EGFRCSF1RACHEBACE1PDE10A
SCHEMBL8648606 1.00 EGFR (0.54) EGFRCSF1RACHEBACE1PDE10A
SCHEMBL8649521 1.00 EGFR (0.54) EGFRCSF1RACHEBACE1PDE10A
SCHEMBL8648604 1.00 EGFR (0.54) EGFRCSF1RACHEBACE1PDE10A
SCHEMBL8647403 0.78 EGFR (0.61) EGFRCSF1RACHEBACE1PDE10A
SCHEMBL4718427 0.76 EGFR (0.65) EGFRCSF1RACHEBACE1PDE10A
Hydrochloric Acid SCHEMBL6181670 0.75 EGFR (0.66) EGFRCSF1RACHEBACE1PDE10A
SCHEMBL27477800 0.74 EGFR (0.60) EGFRCSF1RACHEBACE1PDE10A
SCHEMBL9113385 0.72 EGFR (0.57) EGFRCSF1RACHEBACE1PDE10A
SCHEMBL23721410 0.72 ACHE (0.75) EGFRACHEBACE1PDE10AKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5736534-A HYPERPROLIFERATIVE DISEASES; INHIBITORS OF PROTEIN-TYROSINE KINASES SUCH AS EPIDERMAL GROWTH FACTOR RECEPTOR; BRAIN, LUNG, BREAST CANCER; PSORIASIS AND BENIGN PROSTATE HYPERPLASIA PFIZER INC. (US) 1998-04-07 US disclosed
WO-1995023141-A1 4-HETEROCYCLYL-SUBSTITUTED QUINAZOLINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS ANTI-CANCER AGENTS PFIZER INC. (US) 1995-08-31 WO disclosed