SCHEMBL8648779

SCHEMBL8648779

OCCCc1csc2ccc(F)cc12

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 7/20 0.58
MTNR1B P49286 2/20 0.58
CA2 P00918 1/20 0.50
CYP2A6 P11509 3/20 0.40
MPO P05164 1/20 0.39
SLC6A4 P31645 1/20 0.39
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
MAPT P10636 3/20 0.38
TP53 P04637 2/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5234280 0.84 MTNR1A (0.55) MTNR1AMTNR1BCA2CYP2A6MPO
SCHEMBL8435459 0.84 MTNR1A (0.58) MTNR1AMTNR1BCA2CYP2A6MPO
SCHEMBL6985740 0.84 MTNR1A (0.55) MTNR1AMTNR1BCA2CYP2A6MPO
SCHEMBL2094883 0.81 MTNR1A (0.52) MTNR1AMTNR1BCA2CYP2A6MPO
SCHEMBL23612316 0.81 CYP2A6 (0.41) MTNR1AMTNR1BCYP2A6KEAP1NFE2L2
SCHEMBL8653030 0.81 CYP2A6 (0.61) MTNR1AMTNR1BCA2CYP2A6KEAP1
SCHEMBL8586113 0.80 MTNR1A (0.57) MTNR1AMTNR1BCA2CYP2A6MPO
SCHEMBL8435339 0.80 MTNR1A (0.61) MTNR1AMTNR1BCA2CYP2A6MPO
SCHEMBL27628031 0.80 MTNR1A (0.57) MTNR1AMTNR1BCA2CYP2A6KEAP1
Hydrochloric Acid SCHEMBL7145521 0.79 MTNR1A (0.56) MTNR1AMTNR1BCA2CYP2A6MPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763444-A CENTRAL NERVOUS SYSTEM AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-06-09 US disclosed
EP-0761666-A2 Antidepressant 1-arylalkyl-4-(alkoxypyridinyl)- or 4-(alkoxypyrimidinyl)piperazine derivatives BRISTOL-MYERS SQUIBB COMPANY (US) 1997-03-12 EP disclosed