SCHEMBL8656197

SCHEMBL8656197

COc1ccc(-c2ccc(F)c(F)c2)cc1F

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.56
PTGS2 P35354 8/20 0.54
PDGFRB P09619 2/20 0.54
PDGFRA P16234 2/20 0.54
PTGS1 P23219 4/20 0.53
ERN1 O75460 1/20 0.53
RAB9A P51151 3/20 0.51
NPC1 O15118 2/20 0.51
ALDH1A1 P00352 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
TDP2 O95551 1/20 0.49
LMNA P02545 2/20 0.48
MAPK1 P28482 1/20 0.48
HTT P42858 1/20 0.48
TUBB1 Q9H4B7 1/20 0.47
MGLL Q99685 1/20 0.47
KDM4E B2RXH2 1/20 0.46
MAPT P10636 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9464193 0.93 CYP17A1 (0.61) CYP17A1PTGS2PDGFRBPDGFRAPTGS1
SCHEMBL13906291 0.86 CYP17A1 (0.55) CYP17A1PTGS2PDGFRBPDGFRAPTGS1
SCHEMBL15605813 0.85 CYP17A1 (0.58) CYP17A1PTGS2PDGFRBPDGFRAPTGS1
SCHEMBL6368263 0.84 PTGS2 (0.56) CYP17A1PTGS2PDGFRBPDGFRAPTGS1
SCHEMBL8481713 0.83 CYP17A1 (0.57) CYP17A1PTGS2PDGFRBPDGFRAPTGS1
SCHEMBL19722074 0.83 CYP17A1 (0.57) CYP17A1PTGS2PDGFRBPDGFRAPTGS1
SCHEMBL10093049 0.83 CYP17A1 (0.57) CYP17A1PTGS2PDGFRBPDGFRAPTGS1
SCHEMBL7783072 0.83 CYP17A1 (0.57) CYP17A1PTGS2PDGFRBPDGFRAPTGS1
SCHEMBL17279129 0.82 ERN1 (0.56) CYP17A1PTGS2PDGFRBPDGFRAERN1
SCHEMBL14270106 0.81 TUBB1 (0.49) CYP17A1PTGS2PDGFRBPDGFRAPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7399505-B2 Fluorinated phenanthrenes and their use in liquid-crystal mixtures MERCK PATENT GMBH (DE) 2008-07-15 US disclosed
US-5739166-A ALKYLSULFONYL OR AMINOSULFONYL SUBSTITUTED AROMATIC COMPOUNDS AS NON-STEROIDAL ANTIINFLAMMATORY AGENT G.D. SEARLE & CO. (US) 1998-04-14 US disclosed