SCHEMBL8656275

SCHEMBL8656275

Sn1nncc1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.49
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2C19 P33261 1/20 0.45
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
HDAC1 Q13547 1/20 0.38
FLT3 P36888 3/20 0.38
GSK3B P49841 2/20 0.38
CYP2D6 P10635 1/20 0.37
KCNMA1 Q12791 1/20 0.37
MAPK9 P45984 1/20 0.37
MAPK10 P53779 1/20 0.37
RAC2 P15153 1/20 0.36
RAC3 P60763 1/20 0.36
CDC42 P60953 1/20 0.36
RAC1 P63000 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1395472 0.77 TSHR (0.70) TSHRCYP1A2CYP3A4CYP2C19PTGS1
SCHEMBL11280381 0.74 CYP1A2 (0.45) TSHRCYP1A2CYP3A4CYP2C19PTGS1
SCHEMBL1336097 0.74 CYP1A2 (0.45) TSHRCYP1A2CYP3A4CYP2C19PTGS1
SCHEMBL3320095 0.74 PTGS1 (0.46) TSHRCYP1A2CYP3A4CYP2C19PTGS1
SCHEMBL5326699 0.74 PTGS1 (0.46) TSHRCYP1A2CYP3A4CYP2C19PTGS1
SCHEMBL5139302 0.74 CYP1A2 (0.45) TSHRCYP1A2CYP3A4CYP2C19PTGS1
SCHEMBL8653609 0.71 KEAP1 (0.49) TSHRCYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL8655764 0.70 CYP11B2 (0.46) TSHRALDH1A1IDO1CYP11B2
SCHEMBL24011415 0.69 HDAC1 (0.48) TSHRCYP1A2CYP3A4CYP2C19PTGS1
SCHEMBL2759113 0.69 PTGS1 (0.43) TSHRCYP1A2CYP3A4CYP2C19PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4917995-A CONTAINING COMPOUND CAPABLE OF CHANGING THE TONE OF SILVER IMAGES WITHOUT LOWERING SENSITIVITY FUJI PHOTO FILM CO., LTD. (JP) 1990-04-17 US claimed
EP-0436027-B1 METHOD OF TREATING SILVER HALIDE PHOTOGRAPHIC MATERIAL FUJI PHOTO FILM CO LTD (JP) 1998-10-14 EP disclosed
US-5780198-A MULTILAYER; CONTAINS A HYDRAZINE NUCLEATING AGENT AND A REDOX COMPOUND CAPABLE OF RELEASING A DEVELOPMENT INHIBITOR WHEN THE REDOX COMPOUND IS OXIDIZED; ULTRAHIGH CONTRAST IMAGE WITH BROAD DOT GRADATION FUJI PHOTO FILM CO., LTD. (JP) 1998-07-14 US disclosed
EP-0442323-B1 Silver halide color reversal photographic material capable of providing interimage effect FUJI PHOTO FILM CO LTD (JP) 1997-10-15 EP disclosed
EP-0420005-B1 High contrast silver halide photographic material FUJI PHOTO FILM CO LTD (JP) 1996-07-10 EP disclosed
EP-0395069-B1 Silver halide photographic materials FUJI PHOTO FILM CO LTD (JP) 1996-07-10 EP disclosed
EP-0335319-B1 Silver halide photographic material FUJI PHOTO FILM CO LTD (JP) 1996-06-05 EP disclosed
EP-0398285-B1 Silver halide photographic materials FUJI PHOTO FILM CO LTD (JP) 1995-09-13 EP disclosed
EP-0393720-B1 Silver halide photographic materials FUJI PHOTO FILM CO LTD (JP) 1995-08-23 EP disclosed
US-5395732-A Silver halide photographic materials FUJI PHOTO FILM CO., LTD. (JP) 1995-03-07 US disclosed
EP-0436027-A1 METHOD OF TREATING SILVER HALIDE PHOTOGRAPHIC MATERIAL FUJI PHOTO FILM CO., LTD. (JP) 1991-07-10 EP disclosed
US-5006444-A Silver halide photographic material FUJI PHOTO FILM CO., LTD. (JP) 1991-04-09 US disclosed
EP-0420005-A1 high contrast silver halide photographic material FUJI PHOTO FILM CO., LTD. (JP) 1991-04-03 EP disclosed
EP-0398285-A2 Silver halide photographic materials FUJI PHOTO FILM CO., LTD. (JP) 1990-11-22 EP disclosed
EP-0395069-A2 Silver halide photographic materials FUJI PHOTO FILM CO., LTD. (JP) 1990-10-31 EP disclosed
EP-0393720-A2 Silver halide photographic materials FUJI PHOTO FILM CO., LTD. (JP) 1990-10-24 EP disclosed
US-4917995-A CONTAINING COMPOUND CAPABLE OF CHANGING THE TONE OF SILVER IMAGES WITHOUT LOWERING SENSITIVITY FUJI PHOTO FILM CO., LTD. (JP) 1990-04-17 US disclosed
EP-0335319-A2 Silver halide photographic material FUJI PHOTO FILM CO., LTD. (JP) 1989-10-04 EP disclosed
US-4737442-A INCLUDING A SENSITIZER AND A BLOCKED DEVELOPMENT RESTRAINER; FREE OF BLACK SPOTS FUJI PHOTO FILM CO., LTD. (JP) 1988-04-12 US disclosed
EP-0226953-A2 Color photographic recording material Agfa-Gevaert AG (DE) 1987-07-01 EP disclosed