SCHEMBL8656757

SCHEMBL8656757

COc1cc(OC)cc(-c2c(F)c(F)c(F)c(F)c2-c2ccccc2S(N)(=O)=O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 1/20 0.41
ABL1 P00519 2/20 0.41
ABCB1 P08183 2/20 0.41
BCR P11274 2/20 0.41
P2RX3 P56373 1/20 0.41
MAPT P10636 2/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
USP2 O75604 1/20 0.40
PKM P14618 1/20 0.40
KMT2A Q03164 1/20 0.40
F10 P00742 3/20 0.39
ALOX5AP P20292 4/20 0.39
FEN1 P39748 4/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
P2RY4 P51582 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8661969 0.90 PTGES2 (0.50) PTGES2F10ADORA2AADORA1
SCHEMBL8661361 0.88 MAPT (0.49) MAPTPTGS1KMT2AF10NPC1
SCHEMBL8659866 0.87 PTGS2 (0.45) P2RX3MAPTPTGS1PTGS2USP2
SCHEMBL8660193 0.86 PTGS2 (0.44) PTGES2MAPTPTGS1PTGS2F10
SCHEMBL8661079 0.85 PTGS2 (0.39) MAPTPTGS1PTGS2F10ALOX5AP
SCHEMBL8657401 0.85 PTGS2 (0.43) P2RX3MAPTPTGS1PTGS2USP2
SCHEMBL8657899 0.85 CA9 (0.47) MAPTPTGS1PTGS2KMT2AALOX5AP
SCHEMBL8661477 0.84 PTGS2 (0.54) PTGES2PTGS1PTGS2F10ALOX5AP
SCHEMBL8657860 0.84 PTGS2 (0.43) PTGES2MAPTPTGS1PTGS2USP2
SCHEMBL8660480 0.82 ALOX5AP (0.41) PTGS1PTGS2KMT2AF10ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739166-A ALKYLSULFONYL OR AMINOSULFONYL SUBSTITUTED AROMATIC COMPOUNDS AS NON-STEROIDAL ANTIINFLAMMATORY AGENT G.D. SEARLE & CO. (US) 1998-04-14 US disclosed