SCHEMBL8661079

SCHEMBL8661079

COc1c(C)cc(-c2c(F)c(F)c(F)c(F)c2-c2ccccc2S(N)(=O)=O)cc1C

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.39
PTGS1 P23219 5/20 0.39
ALOX5AP P20292 7/20 0.38
FEN1 P39748 7/20 0.38
ALDH1A1 P00352 1/20 0.36
LCK P06239 1/20 0.36
GLA P06280 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
LIMK1 P53667 1/20 0.36
LIMK2 P53671 1/20 0.36
F10 P00742 1/20 0.35
CA2 P00918 3/20 0.35
CA12 O43570 3/20 0.35
CA9 Q16790 3/20 0.35
CA1 P00915 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8660193 0.89 PTGS2 (0.44) PTGS2PTGS1ALOX5APFEN1ALDH1A1
SCHEMBL8663491 0.88 ALOX5AP (0.41) PTGS2PTGS1ALOX5APFEN1CA2
SCHEMBL8657899 0.88 CA9 (0.47) PTGS2PTGS1ALOX5APFEN1ALDH1A1
SCHEMBL8661432 0.87 ALOX5AP (0.40) PTGS2PTGS1ALOX5APFEN1F10
SCHEMBL8661477 0.86 PTGS2 (0.54) PTGS2PTGS1ALOX5APFEN1F10
SCHEMBL8661468 0.85 PTGS2 (0.56) PTGS2PTGS1ALOX5APFEN1ALDH1A1
SCHEMBL8657401 0.85 PTGS2 (0.43) PTGS2PTGS1ALOX5APFEN1ALDH1A1
SCHEMBL8657919 0.85 PTGS1 (0.39) PTGS2PTGS1ALOX5APFEN1F10
SCHEMBL8656757 0.85 PTGES2 (0.41) PTGS2PTGS1ALOX5APFEN1MAPT
SCHEMBL8659866 0.85 PTGS2 (0.45) PTGS2PTGS1ALOX5APFEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739166-A ALKYLSULFONYL OR AMINOSULFONYL SUBSTITUTED AROMATIC COMPOUNDS AS NON-STEROIDAL ANTIINFLAMMATORY AGENT G.D. SEARLE & CO. (US) 1998-04-14 US disclosed