SCHEMBL8657995

SCHEMBL8657995

COc1cccc(-c2ccccc2NS(=O)(=O)c2ccccc2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 4/20 0.62
PTGES2 Q9H7Z7 1/20 0.62
KEAP1 Q14145 3/20 0.59
NFE2L2 Q16236 2/20 0.59
MCOLN3 Q8TDD5 2/20 0.58
CA12 O43570 1/20 0.58
CA2 P00918 1/20 0.58
LMNA P02545 1/20 0.58
CA9 Q16790 1/20 0.58
TUBB4A P04350 2/20 0.56
TUBB P07437 2/20 0.56
TUBA3C P0DPH7 2/20 0.56
TUBA1B P68363 2/20 0.56
TUBA4A P68366 2/20 0.56
TUBB4B P68371 2/20 0.56
TUBB3 Q13509 2/20 0.56
TUBB2A Q13885 2/20 0.56
TUBB8 Q3ZCM7 2/20 0.56
TUBA3E Q6PEY2 2/20 0.56
TUBA1A Q71U36 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8660187 0.89 STAT3 (0.62) STAT3PTGES2KEAP1NFE2L2MCOLN3
SCHEMBL8649422 0.88 PTGES2 (0.56) STAT3PTGES2KEAP1NFE2L2TUBB4A
SCHEMBL28452095 0.85 SLC22A12 (0.74) STAT3PTGES2KEAP1NFE2L2PGR
SCHEMBL8659936 0.85 STAT3 (0.58) STAT3PTGES2KEAP1NFE2L2TUBB4A
SCHEMBL2518687 0.85 STAT3 (0.80) STAT3KEAP1NFE2L2MCOLN3CA12
SCHEMBL8662980 0.85 STAT3 (0.80) STAT3KEAP1NFE2L2MCOLN3CA12
SCHEMBL21708292 0.83 KEAP1 (0.60) STAT3PTGES2KEAP1NFE2L2MCOLN3
SCHEMBL8660547 0.82 LMNA (0.71) STAT3MCOLN3CA12CA2LMNA
SCHEMBL21708334 0.81 STAT3 (0.57) STAT3PTGES2KEAP1NFE2L2TUBB4A
SCHEMBL8663502 0.81 PTGES2 (0.51) STAT3PTGES2KEAP1NFE2L2TUBB4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739166-A ALKYLSULFONYL OR AMINOSULFONYL SUBSTITUTED AROMATIC COMPOUNDS AS NON-STEROIDAL ANTIINFLAMMATORY AGENT G.D. SEARLE & CO. (US) 1998-04-14 US disclosed