SCHEMBL8658285

SCHEMBL8658285

CC(C)(C)[Si](C)(C)Oc1cc2ccc(-c3cc(C(=O)O)cs3)cc2cc1C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARG P13631 11/20 0.51
RARB P10826 10/20 0.51
RARA P10276 10/20 0.51
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
NR1I2 O75469 1/20 0.51
LMNA P02545 1/20 0.51
PGR P06401 1/20 0.51
HSPD1 P10809 1/20 0.51
GOT1 P17174 1/20 0.51
GLRA1 P23415 1/20 0.51
BLM P54132 1/20 0.51
HSPE1 P61604 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
THRB P10828 1/20 0.48
RECQL P46063 1/20 0.48
NR2E1 Q9Y466 1/20 0.48
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
TP53 P04637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8692906 0.89 RARB (0.41) RARGRARBRARAMEN1KMT2A
SCHEMBL8659574 0.88 RARB (0.63) RARGRARBRARAMEN1KMT2A
SCHEMBL8900640 0.88 MEN1 (0.64) RARGRARBRARAMEN1KMT2A
SCHEMBL981497 0.82 RARG (0.72) RARGRARBRARAMEN1KMT2A
SCHEMBL8656655 0.82 RARG (0.48) RARGRARBRARAMEN1KMT2A
SCHEMBL8657215 0.81 MEN1 (0.72) RARGRARBRARAMEN1KMT2A
SCHEMBL8458638 0.77 RARG (0.55) RARGRARBRARAMEN1KMT2A
SCHEMBL8690840 0.76 RARB (0.51) RARGRARBRARAMEN1KMT2A
SCHEMBL8660077 0.76 RARA (0.38) RARGRARBRARAMEN1KMT2A
SCHEMBL7077371 0.75 RARB (0.61) RARGRARBRARAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0658553-B1 Polycyclic aromatic compounds, pharmaceutical and cosmetic compositions containing them and uses thereof CIRD GALDERMA (FR) 1998-11-04 EP disclosed
EP-0658553-A1 Polycyclic aromatic compounds, pharmaceutical compositions containing them and uses thereof CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA, ( CIRD GALDERMA) (FR) 1995-06-21 EP disclosed