SCHEMBL8659331

SCHEMBL8659331

Cc1cc(Oc2ccc(Br)cc2F)c(Cl)c(C)c1NC(=O)NC(=O)c1ccccc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYGL P06737 5/20 0.46
GCGR P47871 1/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
POLB P06746 3/20 0.40
RAB9A P51151 3/20 0.40
NPC1 O15118 2/20 0.40
TP53 P04637 1/20 0.40
PKM P14618 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
MAPT P10636 4/20 0.37
GAA P10253 1/20 0.37
RECQL P46063 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
PCTP Q9UKL6 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
GHSR Q92847 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8656117 0.91 PYGL (0.48) PYGLGCGRKMT2AMEN1POLB
SCHEMBL8659406 0.87 KMT2A (0.42) PYGLKMT2AMEN1RAB9ANPC1
SCHEMBL9138760 0.87 KMT2A (0.43) KMT2AMEN1POLBPKMTDP1
SCHEMBL8659832 0.86 GCGR (0.49) PYGLGCGRKMT2AMEN1POLB
SCHEMBL8660959 0.85 PYGL (0.47) PYGLGCGRKMT2AMEN1POLB
SCHEMBL8657616 0.85 GCGR (0.48) PYGLGCGRKMT2AMEN1POLB
SCHEMBL8662856 0.84 PYGL (0.46) PYGLGCGRKMT2AMEN1POLB
SCHEMBL8658826 0.84 KMT2A (0.47) PYGLKMT2AMEN1RAB9ANPC1
SCHEMBL8657591 0.84 GCGR (0.56) PYGLGCGRKMT2AMEN1POLB
SCHEMBL8673485 0.84 KMT2A (0.54) PYGLGCGRKMT2AMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed