SCHEMBL8656117

SCHEMBL8656117

Cc1cc(Oc2ccc(Br)cc2Br)c(Cl)c(C)c1NC(=O)NC(=O)c1ccccc1Cl

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PYGL P06737 3/20 0.48
GCGR P47871 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
POLB P06746 3/20 0.41
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.41
PKM P14618 1/20 0.41
MAPT P10636 5/20 0.39
GAA P10253 1/20 0.39
RECQL P46063 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
PCTP Q9UKL6 1/20 0.38
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
GHSR Q92847 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8655824 0.92 PYGL (0.48) PYGLGCGRMEN1KMT2APOLB
SCHEMBL8657616 0.92 GCGR (0.48) PYGLGCGRMEN1KMT2APOLB
SCHEMBL8660959 0.91 PYGL (0.47) PYGLGCGRMEN1KMT2APOLB
SCHEMBL8659406 0.91 KMT2A (0.42) PYGLMEN1KMT2ARAB9ANPC1
SCHEMBL8659331 0.91 PYGL (0.46) PYGLGCGRMEN1KMT2APOLB
SCHEMBL8660844 0.89 MAPT (0.41) PYGLMEN1KMT2APOLBRAB9A
SCHEMBL8662856 0.89 PYGL (0.46) PYGLGCGRMEN1KMT2APOLB
SCHEMBL8660840 0.88 MAPT (0.40) PYGLMEN1KMT2APOLBRAB9A
SCHEMBL8659728 0.87 PYGL (0.49) PYGLGCGRKMT2APOLBRAB9A
SCHEMBL8661424 0.85 GCGR (0.49) PYGLGCGRMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed