SCHEMBL8659337

SCHEMBL8659337

CCCC1(CCC)CCSc2ccc(C#Cc3ccccc3C(=O)O)cc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 10/20 0.46
RARG P13631 10/20 0.46
RARA P10276 9/20 0.46
CYP3A4 P08684 3/20 0.43
CYP26A1 O43174 2/20 0.43
KMT2A Q03164 1/20 0.40
FFAR1 O14842 6/20 0.35
CRABP2 P29373 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
HNF4A P41235 1/20 0.33
FFAR4 Q5NUL3 2/20 0.33
RXRA P19793 1/20 0.32
CHRM2 P08172 1/20 0.32
S1PR1 P21453 1/20 0.32
FPR1 P21462 1/20 0.32
FPR3 P25089 1/20 0.32
GPR183 P32249 1/20 0.32
APLNR P35414 1/20 0.32
GPR65 Q8IYL9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7654860 0.84 CYP3A4 (0.54) RARBRARGRARACYP3A4CYP26A1
SCHEMBL27304274 0.84 RARB (0.62) RARBRARGRARACYP3A4CYP26A1
SCHEMBL7648981 0.76 RARB (0.61) RARBRARGRARACYP3A4CYP26A1
SCHEMBL7654342 0.76 CYP3A4 (0.53) RARBRARGRARACYP3A4CYP26A1
SCHEMBL9817722 0.76 RARA (0.63) RARBRARGRARACYP3A4CYP26A1
SCHEMBL7650773 0.74 RARA (0.40) RARBRARGRARACYP3A4CYP26A1
SCHEMBL7650870 0.74 CYP3A4 (0.35) RARBRARGRARACYP3A4CYP26A1
SCHEMBL8580705 0.72 RARB (0.65) RARBRARGRARACYP3A4CYP26A1
SCHEMBL8037152 0.71 RARA (0.52) RARBRARGRARACYP3A4CYP26A1
SCHEMBL7659037 0.71 CYP3A4 (0.46) RARBRARGRARACYP3A4CYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750693-A THIOCHROMANYL OR CHROMANYL COMPOUNDS AS ANTICARCINOGINIC AGENTS, SKIN DISORDERS AND ATHEROSCLEROSIS ALLERGAN (US) 1998-05-12 US disclosed
US-5677451-A CONTROLLING CELL DIFFERENTIATION; SKIN DISORDERS; ANTICANCER AGENTS ALLERGAN (US) 1997-10-14 US disclosed