SCHEMBL8659474

SCHEMBL8659474

Cc1cc(N(c2ccccc2)S(=O)(=O)c2ccccc2)ccc1N(C)C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.50
ESR1 P03372 1/20 0.47
ALDH1A1 P00352 2/20 0.45
NPSR1 Q6W5P4 2/20 0.43
MAPT P10636 1/20 0.43
CA12 O43570 1/20 0.43
CA9 Q16790 1/20 0.43
HTR6 P50406 1/20 0.41
KMT2A Q03164 1/20 0.40
NR1I2 O75469 1/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
CNR2 P34972 1/20 0.38
HTT P42858 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
C5AR1 P21730 1/20 0.37
LMNA P02545 1/20 0.37
GBA1 P04062 1/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8660081 0.88 PKM (0.50) PKMESR1ALDH1A1NPSR1MAPT
SCHEMBL8656891 0.84 PKM (0.49) PKMESR1ALDH1A1CA12CA9
SCHEMBL8660463 0.84 PKM (0.49) PKMESR1ALDH1A1MAPTCA12
SCHEMBL8663426 0.83 PKM (0.45) PKMESR1ALDH1A1NPSR1MAPT
SCHEMBL8660142 0.83 PKM (0.54) PKMESR1ALDH1A1NPSR1MAPT
SCHEMBL8663371 0.82 PKM (0.53) PKMESR1ALDH1A1CA12CA9
SCHEMBL8662811 0.82 PKM (0.46) PKMESR1ALDH1A1NPSR1KEAP1
SCHEMBL8662966 0.81 PKM (0.49) PKMESR1ALDH1A1MAPTCA12
SCHEMBL8658102 0.81 PKM (0.49) PKMESR1ALDH1A1CA12CA9
SCHEMBL8656925 0.81 PKM (0.63) PKMESR1ALDH1A1CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739166-A ALKYLSULFONYL OR AMINOSULFONYL SUBSTITUTED AROMATIC COMPOUNDS AS NON-STEROIDAL ANTIINFLAMMATORY AGENT G.D. SEARLE & CO. (US) 1998-04-14 US disclosed