SCHEMBL8658102

SCHEMBL8658102

CN(C)c1cc(N(c2ccccc2)S(=O)(=O)c2ccccc2)ccc1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.49
ESR1 P03372 1/20 0.46
ALDH1A1 P00352 2/20 0.41
PSEN1 P49768 1/20 0.40
PSEN2 P49810 1/20 0.40
APH1B Q8WW43 1/20 0.40
NCSTN Q92542 1/20 0.40
APH1A Q96BI3 1/20 0.40
PSENEN Q9NZ42 1/20 0.40
HTR6 P50406 1/20 0.40
KMT2A Q03164 3/20 0.39
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
NR1H3 Q13133 2/20 0.39
APOBEC3G Q9HC16 1/20 0.39
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
HSD17B10 Q99714 1/20 0.38
NR1H2 P55055 2/20 0.38
FFAR1 O14842 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8656891 0.89 PKM (0.49) PKMESR1ALDH1A1HTR6KMT2A
SCHEMBL8658024 0.85 PKM (0.51) PKMESR1ALDH1A1HTR6KMT2A
SCHEMBL8660081 0.84 PKM (0.50) PKMESR1ALDH1A1HTR6KMT2A
SCHEMBL8662966 0.83 PKM (0.49) PKMESR1ALDH1A1HTR6KMT2A
SCHEMBL8661181 0.82 PKM (0.45) PKMESR1ALDH1A1HTR6KMT2A
SCHEMBL8659474 0.81 PKM (0.50) PKMESR1ALDH1A1HTR6KMT2A
SCHEMBL8663371 0.81 PKM (0.53) PKMESR1ALDH1A1HTR6KMT2A
SCHEMBL8659118 0.81 PKM (0.53) PKMESR1ALDH1A1HTR6KMT2A
SCHEMBL8660320 0.81 PKM (0.46) PKMESR1ALDH1A1KMT2AMAPK1
SCHEMBL8660463 0.80 PKM (0.49) PKMESR1ALDH1A1HTR6KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739166-A ALKYLSULFONYL OR AMINOSULFONYL SUBSTITUTED AROMATIC COMPOUNDS AS NON-STEROIDAL ANTIINFLAMMATORY AGENT G.D. SEARLE & CO. (US) 1998-04-14 US disclosed