SCHEMBL8659481

SCHEMBL8659481

CCCC(=O)Oc1ccc(C#Cc2ccc3c(c2)C(SCC)(SCC)CCO3)o1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 5/20 0.34
PRSS2 P07478 5/20 0.34
PRSS3 P35030 5/20 0.34
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
HPGD P15428 1/20 0.31
AKR1B1 P15121 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8658357 0.93 ALDH1A1 (0.33) PRSS1PRSS2PRSS3
SCHEMBL8661596 0.85
SCHEMBL8664184 0.83 CYP3A4 (0.33) HPGD
SCHEMBL8661981 0.82 HPGD (0.30) HPGD
SCHEMBL8662239 0.81 CYP3A4 (0.35)
SCHEMBL8662230 0.80 CYP3A4 (0.36)
SCHEMBL7652315 0.80 CYP26A1 (0.37) PRSS1PRSS2PRSS3MAOAMAOB
SCHEMBL8671496 0.75 KMT2A (0.45) MAOAHPGD
SCHEMBL8659480 0.74 CYP3A4 (0.40)
SCHEMBL7817655 0.74 ACACB (0.32) AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750693-A THIOCHROMANYL OR CHROMANYL COMPOUNDS AS ANTICARCINOGINIC AGENTS, SKIN DISORDERS AND ATHEROSCLEROSIS ALLERGAN (US) 1998-05-12 US disclosed
US-5677451-A CONTROLLING CELL DIFFERENTIATION; SKIN DISORDERS; ANTICANCER AGENTS ALLERGAN (US) 1997-10-14 US disclosed