SCHEMBL8659667

SCHEMBL8659667

O=C(NC(=O)c1ccccc1Cl)Nc1ccc(Oc2ccc(C(F)(F)F)c(Cl)n2)c(Cl)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GCGR P47871 1/20 0.60
TDP1 Q9NUW8 1/20 0.51
PNLIP P16233 2/20 0.48
S1PR1 P21453 4/20 0.46
STK39 Q9UEW8 1/20 0.46
PLCG2 P16885 1/20 0.46
POLB P06746 2/20 0.45
NPC1 O15118 1/20 0.45
PKM P14618 1/20 0.45
RAB9A P51151 1/20 0.45
KDR P35968 2/20 0.45
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
GRM4 Q14833 2/20 0.44
PYGL P06737 1/20 0.43
BRAF P15056 1/20 0.43
MAPK14 Q16539 1/20 0.43
TNNI3K Q59H18 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11249648 0.94 GCGR (0.52) GCGRTDP1PNLIPS1PR1STK39
SCHEMBL11239027 0.93 GCGR (0.51) GCGRTDP1S1PR1PLCG2POLB
SCHEMBL11246898 0.93 PNLIP (0.52) GCGRTDP1PNLIPS1PR1STK39
SCHEMBL11256445 0.92 GCGR (0.50) GCGRTDP1S1PR1PLCG2POLB
SCHEMBL11244163 0.92 PNLIP (0.51) GCGRTDP1PNLIPS1PR1STK39
SCHEMBL11248306 0.92 PNLIP (0.51) GCGRTDP1PNLIPS1PR1STK39
SCHEMBL11245283 0.92 GCGR (0.50) GCGRTDP1PNLIPS1PR1STK39
SCHEMBL11248757 0.92 GCGR (0.59) GCGRTDP1PNLIPS1PR1STK39
SCHEMBL11256032 0.91 GCGR (0.58) GCGRTDP1PNLIPS1PR1STK39
SCHEMBL11247233 0.89 GCGR (0.47) GCGRS1PR1STK39POLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4321388-A N-benzoyl N'-pyridyloxy phenyl urea ISHIHARA SANGYO KAISHA LTD. (JP) 1982-03-23 US claimed
EP-0025363-A1 N-Benzoyl N'-pyridyloxy phenyl ureas, a process for their production and pharmaceutical and insecticidal compositions containing the same ISHIHARA SANGYO KAISHA LTD. (JP) 1981-03-18 EP claimed
JP-62005959-A None JP disclosed
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
JP-S625959-A BENZOYLUREA COMPOUND ISHIHARA SANGYO KAISHA LTD 1987-01-12 JP disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed
EP-0025363-B1 N-BENZOYL N'-PYRIDYLOXY PHENYL UREAS, A PROCESS FOR THEIR PRODUCTION AND PHARMACEUTICAL AND INSECTICIDAL COMPOSITIONS CONTAINING THE SAME ISHIHARA SANGYO KAISHA LTD. (JP) 1982-08-25 EP disclosed
US-4321388-A N-benzoyl N'-pyridyloxy phenyl urea ISHIHARA SANGYO KAISHA LTD. (JP) 1982-03-23 US disclosed
EP-0025363-A1 N-Benzoyl N'-pyridyloxy phenyl ureas, a process for their production and pharmaceutical and insecticidal compositions containing the same ISHIHARA SANGYO KAISHA LTD. (JP) 1981-03-18 EP disclosed