SCHEMBL8660859

SCHEMBL8660859

Cc1cc(NC(=O)NC(=O)c2ccccc2Cl)cc(C)c1Oc1ccc(Cl)c2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESRRA P11474 5/20 0.53
GCGR P47871 1/20 0.53
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
POLB P06746 1/20 0.50
PKM P14618 1/20 0.50
PYGL P06737 4/20 0.49
TDP1 Q9NUW8 1/20 0.46
PCTP Q9UKL6 1/20 0.45
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ATM Q13315 1/20 0.43
PLCG2 P16885 1/20 0.43
PNLIP P16233 1/20 0.41
TP53 P04637 1/20 0.41
KIT P10721 1/20 0.41
PDGFRA P16234 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10963721 0.96 ESRRA (0.54) ESRRAGCGRNPC1RAB9APOLB
SCHEMBL8659992 0.91 ESRRA (0.47) ESRRAGCGRNPC1RAB9APOLB
SCHEMBL8655821 0.90 GCGR (0.58) ESRRAGCGRNPC1RAB9APOLB
SCHEMBL8660966 0.89 ESRRA (0.58) ESRRAGCGRNPC1RAB9APOLB
SCHEMBL8656589 0.86 ESRRA (0.45) ESRRAGCGRNPC1RAB9APYGL
SCHEMBL8657108 0.86 PYGL (0.51) ESRRAGCGRNPC1RAB9APOLB
SCHEMBL9133702 0.85 ESRRA (0.46) ESRRANPC1RAB9APOLBMEN1
SCHEMBL8659953 0.85 ESRRA (0.47) ESRRANPC1RAB9APOLBPKM
SCHEMBL10959798 0.85 GCGR (0.50) GCGRNPC1RAB9APOLBPKM
SCHEMBL10963372 0.84 PYGL (0.58) ESRRAGCGRNPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0050321-B1 NOVEL BICYCLOOXYPHENYL UREAS, PROCESS FOR THEIR PREPARATION AND PESTICIDES CONTAINING THEM UNION CARBIDE CORPORATION (US) 1985-08-21 EP claimed
US-4426385-A Insecticidal bicyclooxyphenyl ureas UNION CARBIDE CORPORATION (US) 1984-01-17 US claimed
EP-0050321-A2 Novel bicyclooxyphenyl ureas, process for their preparation and pesticides containing them UNION CARBIDE CORPORATION (US) 1982-04-28 EP claimed
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed
EP-0050321-B1 NOVEL BICYCLOOXYPHENYL UREAS, PROCESS FOR THEIR PREPARATION AND PESTICIDES CONTAINING THEM UNION CARBIDE CORPORATION (US) 1985-08-21 EP disclosed
US-4426385-A Insecticidal bicyclooxyphenyl ureas UNION CARBIDE CORPORATION (US) 1984-01-17 US disclosed
EP-0050321-A2 Novel bicyclooxyphenyl ureas, process for their preparation and pesticides containing them UNION CARBIDE CORPORATION (US) 1982-04-28 EP disclosed