SCHEMBL8660905

SCHEMBL8660905

CCc1cc(C#Cc2ccc3c(c2)C(CC)(CC)CCS3)nnc1CCCCC(=O)O

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RARA P10276 2/20 0.43
RARB P10826 2/20 0.43
RARG P13631 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP26A1 O43174 1/20 0.43
KMT2A Q03164 1/20 0.42
FFAR1 O14842 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8865750 0.81 RARA (0.41) RARARARBRARGCYP3A4CYP26A1
SCHEMBL7653882 0.78 CYP3A4 (0.49) RARARARBRARGCYP3A4CYP26A1
SCHEMBL7658980 0.77 CYP3A4 (0.50) RARARARBRARGCYP3A4CYP26A1
SCHEMBL8037152 0.76 RARA (0.52) RARARARBRARGCYP3A4CYP26A1
SCHEMBL7656131 0.74 CYP3A4 (0.53) RARARARBRARGCYP3A4CYP26A1
SCHEMBL7653775 0.74 CYP3A4 (0.57) RARARARBRARGCYP3A4CYP26A1
SCHEMBL9301486 0.73 RARB (0.56) RARARARBRARGCYP3A4CYP26A1
SCHEMBL8662237 0.73 CYP3A4 (0.47) RARARARBRARGCYP3A4CYP26A1
SCHEMBL8671034 0.73 CYP3A4 (0.51) RARARARBRARGCYP3A4CYP26A1
SCHEMBL9301895 0.72 CYP3A4 (0.59) RARARARBRARGCYP3A4CYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750693-A THIOCHROMANYL OR CHROMANYL COMPOUNDS AS ANTICARCINOGINIC AGENTS, SKIN DISORDERS AND ATHEROSCLEROSIS ALLERGAN (US) 1998-05-12 US disclosed
US-5677451-A CONTROLLING CELL DIFFERENTIATION; SKIN DISORDERS; ANTICANCER AGENTS ALLERGAN (US) 1997-10-14 US disclosed