SCHEMBL8663441

SCHEMBL8663441

CCOC(=O)Cc1ccc(C#Cc2cc3c(cc2C)SCCC3(CC)CC)o1

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.32
RARA P10276 1/20 0.32
RARB P10826 1/20 0.32
RARG P13631 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8661600 0.93 CYP3A4 (0.32) CYP3A4RARARARBRARGKMT2A
SCHEMBL7650601 0.90
SCHEMBL7648967 0.89 CYP4Z1 (0.32) CYP3A4RARARARBRARGKMT2A
SCHEMBL8661860 0.87 PPARG (0.32)
SCHEMBL8659483 0.86 CYP3A4 (0.45) CYP3A4RARARARBRARGKMT2A
SCHEMBL8658185 0.83 NPC1 (0.31)
SCHEMBL8664824 0.83 CYP3A4 (0.33) CYP3A4RARARARBRARGKMT2A
SCHEMBL8674063 0.82 FDFT1 (0.40) CYP3A4RARARARBRARGKMT2A
SCHEMBL7655963 0.82 CYP4F2 (0.33) CYP3A4RARARARBRARGKMT2A
SCHEMBL7655266 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750693-A THIOCHROMANYL OR CHROMANYL COMPOUNDS AS ANTICARCINOGINIC AGENTS, SKIN DISORDERS AND ATHEROSCLEROSIS ALLERGAN (US) 1998-05-12 US disclosed
US-5677451-A CONTROLLING CELL DIFFERENTIATION; SKIN DISORDERS; ANTICANCER AGENTS ALLERGAN (US) 1997-10-14 US disclosed