SCHEMBL8664824

SCHEMBL8664824

CCOC(=O)Cc1ccc(C#Cc2cc3c(cc2C)SCCC3(CC)CC)s1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.33
RARA P10276 1/20 0.33
RARB P10826 1/20 0.33
RARG P13631 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8659645 0.93 CYP3A4 (0.33) CYP3A4RARARARBRARGKMT2A
SCHEMBL7657120 0.90 FFAR1 (0.31)
SCHEMBL7651231 0.89 CYP4F2 (0.32) CYP3A4RARARARBRARGKMT2A
SCHEMBL8660140 0.87 AKT1 (0.31)
SCHEMBL8661983 0.86 CYP3A4 (0.46) CYP3A4RARARARBRARGKMT2A
SCHEMBL8674063 0.83 FDFT1 (0.40) CYP3A4RARARARBRARGKMT2A
SCHEMBL8663441 0.83 CYP3A4 (0.32) CYP3A4RARARARBRARGKMT2A
SCHEMBL7651219 0.81 CYP4F2 (0.34) CYP3A4RARARARBRARGKMT2A
SCHEMBL7657246 0.81 FFAR1 (0.34)
SCHEMBL8659849 0.81 CYP3A4 (0.39) CYP3A4RARARARBRARGKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750693-A THIOCHROMANYL OR CHROMANYL COMPOUNDS AS ANTICARCINOGINIC AGENTS, SKIN DISORDERS AND ATHEROSCLEROSIS ALLERGAN (US) 1998-05-12 US disclosed
US-5677451-A CONTROLLING CELL DIFFERENTIATION; SKIN DISORDERS; ANTICANCER AGENTS ALLERGAN (US) 1997-10-14 US disclosed