SCHEMBL8664327

SCHEMBL8664327

Nc1ccc(COC[C@H]2O[C@@H](n3cnc4c(N)ncnc43)[C@H](O)[C@@H]2O)cc1I

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.58
P2RY1 P47900 4/20 0.58
SMN1; SMN2 Q16637 3/20 0.58
P2RY2 P41231 3/20 0.58
SRC P12931 2/20 0.58
DNPH1 O43598 1/20 0.58
PRKAB2 O43741 1/20 0.58
TRPM2 O94759 1/20 0.58
LDHA P00338 1/20 0.58
ADRB2 P07550 1/20 0.58
FBP1 P09467 1/20 0.58
PRKAG1 P54619 1/20 0.58
PRKAA2 P54646 1/20 0.58
PDE4D Q08499 1/20 0.58
KCNH2 Q12809 1/20 0.58
PRKAA1 Q13131 1/20 0.58
PDE3A Q14432 1/20 0.58
TAS1R3 Q7RTX0 1/20 0.58
TAS1R1 Q7RTX1 1/20 0.58
P2RY11 Q96G91 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7860970 0.91 ADORA1 (0.57) ADORA1P2RY1SMN1; SMN2P2RY2SRC
SCHEMBL5356782 0.88 ADORA3 (0.65) ADORA1P2RY1SMN1; SMN2P2RY2SRC
SCHEMBL13268725 0.87 ADORA1 (0.60) ADORA1P2RY1SMN1; SMN2P2RY2SRC
SCHEMBL62486 0.87 ADORA1 (0.65) ADORA1P2RY1SMN1; SMN2P2RY2SRC
SCHEMBL932846 0.87 ADORA1 (0.65) ADORA1P2RY1SMN1; SMN2P2RY2SRC
SCHEMBL13269066 0.85 ADORA1 (0.60) ADORA1P2RY1SMN1; SMN2P2RY2SRC
SCHEMBL13834596 0.85 ADORA1 (0.60) ADORA1P2RY1SMN1; SMN2P2RY2SRC
SCHEMBL13269154 0.85 PDE2A (0.66) ADORA1P2RY1SMN1; SMN2P2RY2SRC
SCHEMBL4541368 0.85 ADORA1 (0.64) ADORA1P2RY1SMN1; SMN2P2RY2SRC
SCHEMBL13269088 0.85 ADORA1 (0.62) ADORA1P2RY1SMN1; SMN2P2RY2SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773423-A XANTHINE RIBOSIDES THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1998-06-30 US disclosed
EP-0689405-A4 METHODS FOR PROTECTING TISSUES AND ORGANS FROM ISCHEMIC DAMAGE GENSIA INC (US) 1996-09-11 EP disclosed
EP-0689405-A1 METHODS FOR PROTECTING TISSUES AND ORGANS FROM ISCHEMIC DAMAGE GENSIA, INC. (US) 1996-01-03 EP disclosed
WO-1994021195-A1 METHODS FOR PROTECTING TISSUES AND ORGANS FROM ISCHEMIC DAMAGE GENSIA, INC. (US) 1994-09-29 WO disclosed