SCHEMBL8664802

SCHEMBL8664802

CC(=O)c1ccc(OC(F)(F)F)cc1Br

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
GAA P10253 2/20 0.48
POLB P06746 1/20 0.48
THRB P10828 1/20 0.48
HPGD P15428 2/20 0.45
CYP3A4 P08684 1/20 0.45
MAPK1 P28482 1/20 0.45
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
EPHX2 P34913 1/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
TGM2 P21980 1/20 0.41
DYRK1A Q13627 1/20 0.41
PIM1 P11309 1/20 0.40
TRPV1 Q8NER1 2/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30294755 0.85 ALDH1A1 (0.50) ALDH1A1GAAPOLBTHRBHPGD
SCHEMBL3030351 0.85 ALDH1A1 (0.52) ALDH1A1GAAPOLBTHRBEPHX2
SCHEMBL15512481 0.83 GAA (0.48) ALDH1A1GAAPOLBTHRBHPGD
SCHEMBL27719541 0.83 THRB (0.45) ALDH1A1GAAPOLBTHRBNPC1
SCHEMBL2317882 0.82 KMT2A (0.52) ALDH1A1HPGDCYP3A4MAPK1NPC1
SCHEMBL17766955 0.81 MAOB (0.54) ALDH1A1HPGDCYP3A4MAPK1EPHX2
SCHEMBL30557826 0.81 MAOB (0.54) ALDH1A1HPGDCYP3A4MAPK1EPHX2
SCHEMBL2325383 0.81 ALDH1A1 (0.64) ALDH1A1HPGDCYP3A4MAPK1NPC1
SCHEMBL30601548 0.80 ALDH1A1 (0.67) ALDH1A1GAAHPGDCYP3A4MAPK1
SCHEMBL898467 0.80 ALDH1A1 (0.67) ALDH1A1GAAHPGDCYP3A4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1167687-C Arylpyridazinones as prostaglandin endoperoxide H synthase biosynthesis inhibitors ���Ͽع����޹�˾ 2004-09-22 CN disclosed
CN-1277605-A Arylpyridazinones as prostaglandin endoperoxide H synthase biosynthesis inhibitors ABBOTT LAB (US) 2000-12-20 CN disclosed
EP-0881220-A1 DIARYLSULTAM DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 1998-12-02 EP disclosed