SCHEMBL8665462

SCHEMBL8665462

COc1cc(OC2CCN(C(C)=O)CC2)ccc1C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OXTR P30559 3/20 0.55
ALDH1A1 P00352 2/20 0.55
AVPR2 P30518 1/20 0.55
AVPR1A P37288 1/20 0.55
HIF1A Q16665 1/20 0.47
PDE4B Q07343 1/20 0.46
QDPR P09417 1/20 0.46
POLB P06746 1/20 0.46
TP53 P04637 1/20 0.45
IKBKB O14920 2/20 0.45
HRH3 Q9Y5N1 1/20 0.44
HRH1 P35367 1/20 0.44
CCR3 P51677 1/20 0.44
CHUK O15111 1/20 0.44
HSD11B1 P28845 1/20 0.44
CYP4F2 P78329 1/20 0.44
CYP4A11 Q02928 1/20 0.44
IGF1R P08069 1/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8669740 0.89 OXTR (0.55) OXTRALDH1A1AVPR2AVPR1AHIF1A
SCHEMBL7355186 0.85 GPR119 (0.54) ALDH1A1PDE4BHRH3
SCHEMBL12311795 0.85 OXTR (0.50) OXTRALDH1A1AVPR2AVPR1APDE4B
SCHEMBL13362079 0.84 OXTR (0.49) OXTRALDH1A1AVPR2AVPR1APDE4B
SCHEMBL8902641 0.83 HIF1A (0.63) ALDH1A1HIF1APDE4B
SCHEMBL7399421 0.82 PDE4B (0.47) OXTRALDH1A1AVPR2AVPR1APDE4B
SCHEMBL12311796 0.82 POLB (0.52) OXTRALDH1A1AVPR2AVPR1APDE4B
SCHEMBL8664983 0.82 OXTR (0.57) OXTRALDH1A1AVPR2AVPR1APDE4B
SCHEMBL16991926 0.81 HIF1A (0.46) OXTRALDH1A1AVPR2AVPR1AHIF1A
SCHEMBL7402370 0.81 PDE4B (0.52) ALDH1A1PDE4BHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756504-A TREATMENT OF DYSMENORRHEA, PREVENTION OF PREMATURE LABOR MERCK & CO., INC. (US) 1998-05-26 US disclosed
EP-0751773-A4 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 1997-07-16 EP disclosed
EP-0751773-A1 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO. INC. (US) 1997-01-08 EP disclosed
US-5464788-A Stopping labor MERCK & CO., INC. (US) 1995-11-07 US disclosed
WO-1995025443-A1 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1995-09-28 WO disclosed