SCHEMBL8666366

SCHEMBL8666366

CCOC(=O)c1csc(C(=O)C(CCCNS(=O)(=O)c2cccc3ccccc23)NC(=N)N)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.45
CTSK P43235 1/20 0.43
SCN1A P35498 2/20 0.41
SCN2A Q99250 2/20 0.41
SCN3A Q9NY46 2/20 0.41
KDM4E B2RXH2 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CNR2 P34972 1/20 0.39
NPY5R Q15761 5/20 0.39
RAB9A P51151 3/20 0.38
NPC1 O15118 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7377699 0.89 CTSK (0.40) HDAC6CTSKKDM4ECNR2NPY5R
SCHEMBL7377692 0.89 CTSK (0.40) HDAC6CTSKKDM4ECNR2NPY5R
SCHEMBL7377703 0.83 CTSK (0.40) HDAC6CTSKCNR2CCR3
SCHEMBL7380912 0.81 F2 (0.43)
SCHEMBL7380915 0.81 F2 (0.43)
SCHEMBL7377714 0.76 CTSK (0.42) HDAC6CTSKKDM4EALDH1A1RAB9A
SCHEMBL4965135 0.75 SMN1; SMN2 (0.55) KDM4ECYP1A2CYP2C19ALDH1A1CYP2C9
SCHEMBL7380919 0.74 F2 (0.43)
SCHEMBL6978879 0.74 CTSK (0.50) HDAC6CTSKKDM4ECYP1A2CYP2C19
SCHEMBL11629096 0.68 SCN1A (0.60) HDAC6SCN1ASCN2ASCN3AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5827860-A Peptidyl heterocycles useful in the treatment of thrombin related disorders ORTHO PHARMACEUTICAL CORPORATION (US) 1998-10-27 US claimed