SCHEMBL6978879

SCHEMBL6978879

CCOC(=O)c1csc(C(=O)C(CCCNC(=O)[C@@H]2CCCN2)NC(=N)N)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.50
SMN1; SMN2 Q16637 3/20 0.42
PRCP P42785 3/20 0.40
CYP1A2 P05177 1/20 0.37
CYP2C19 P33261 1/20 0.37
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
HDAC6 Q9UBN7 1/20 0.34
GAA P10253 1/20 0.34
DPP7 Q9UHL4 1/20 0.34
KDM4E B2RXH2 1/20 0.33
HSP90AA1 P07900 1/20 0.33
TLR2 O60603 1/20 0.33
CCNK O75909 1/20 0.33
CDK12 Q9NYV4 1/20 0.33
PLA2G4A P47712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981100 0.88 PRCP (0.40) CTSKPRCPMEN1KMT2ADPP7
SCHEMBL27491105 0.83 CTSK (0.48) CTSKSMN1; SMN2CYP1A2CYP2C19NPC1
SCHEMBL6972556 0.76
SCHEMBL6979220 0.76 NPC1 (0.41) SMN1; SMN2NPC1RAB9AALDH1A1HSP90AA1
SCHEMBL6970503 0.76 PRCP (0.39) PRCPHDAC6DPP7KDM4ECCNK
SCHEMBL6976548 0.76 MAOA (0.46) SMN1; SMN2CYP1A2NPC1RAB9AMAPT
SCHEMBL6976777 0.74 MAOB (0.43) MAPT
SCHEMBL8666366 0.74 HDAC6 (0.45) CTSKSMN1; SMN2CYP1A2CYP2C19NPC1
SCHEMBL6976622 0.74 SMYD3 (0.41) SMN1; SMN2CYP1A2CYP2C19NPC1RAB9A
SCHEMBL6976837 0.73 F2 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0833839-B1 PEPTIDYL HETEROCYCLES USEFUL IN THE TREATMENT OF THROMBIN RELATED DISORDERS ORTHO PHARMA CORP (US) 2003-01-08 EP claimed