SCHEMBL8666499

SCHEMBL8666499

O=C(NC(=O)c1c(F)cccc1Cl)Nc1cc(Cl)c(Oc2ccc(Cl)cc2)c(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.52
NPC1 O15118 1/20 0.52
ALDH1A1 P00352 1/20 0.52
MAPK1 P28482 1/20 0.52
GCGR P47871 1/20 0.52
TLR8 Q9NR97 7/20 0.51
TLR7 Q9NYK1 3/20 0.51
GAA P10253 3/20 0.50
PNLIP P16233 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
PPIA P62937 1/20 0.45
JAK2 O60674 1/20 0.44
JAK1 P23458 1/20 0.44
TYK2 P29597 1/20 0.44
STK39 Q9UEW8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4152345 0.95 MEN1 (0.51) KDM4ENPC1ALDH1A1MAPK1GCGR
SCHEMBL8657651 0.90 GCGR (0.47) KDM4ENPC1ALDH1A1MAPK1GCGR
SCHEMBL10919264 0.89 GCGR (0.45) KDM4ENPC1ALDH1A1MAPK1GCGR
SCHEMBL10896474 0.89 GCGR (0.45) KDM4ENPC1ALDH1A1MAPK1GCGR
SCHEMBL9683664 0.87 MEN1 (0.52) KDM4ENPC1ALDH1A1MAPK1GCGR
SCHEMBL10943518 0.87 GCGR (0.70) KDM4ENPC1ALDH1A1MAPK1GCGR
SCHEMBL9134026 0.86 ENPP1 (0.48) KDM4ENPC1ALDH1A1MAPK1GCGR
SCHEMBL9135290 0.86 ENPP1 (0.48) KDM4ENPC1ALDH1A1MAPK1GCGR
SCHEMBL8658796 0.85 PNLIP (0.62) NPC1GCGRTLR8PNLIPPPIA
SCHEMBL8662609 0.85 TLR8 (0.54) KDM4ENPC1ALDH1A1MAPK1TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed