SCHEMBL8667664

SCHEMBL8667664

COC(=O)C(NC(=O)OC(C)(C)C)c1ccc(CC(=O)O)cc1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSS P25774 5/20 0.49
CTSK P43235 5/20 0.49
KLK5 Q9Y337 2/20 0.42
PPARA Q07869 6/20 0.41
PPARG P37231 5/20 0.41
ATM Q13315 2/20 0.41
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
PPARD Q03181 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8667675 0.90 CTSS (0.46) CTSSCTSKKLK5PPARAPPARG
SCHEMBL31724481 0.86 CTSS (0.48) CTSSCTSKKLK5PPARAPPARG
SCHEMBL1095762 0.83 CTSK (0.63) CTSSCTSKKLK5ATM
SCHEMBL1951343 0.83 CTSK (0.63) CTSSCTSKKLK5ATM
SCHEMBL1095763 0.83 CTSK (0.63) CTSSCTSKKLK5ATM
SCHEMBL1686961 0.82 CTSS (0.49) CTSSCTSKKLK5PPARAPPARG
SCHEMBL8666252 0.82 MAPT (0.45) CTSSCTSKKLK5PPARAPPARG
SCHEMBL21787641 0.82 CYP4A11 (0.46) CTSSCTSKKLK5PPARAPPARG
SCHEMBL1554126 0.82 CTSS (0.48) CTSSCTSKKLK5
SCHEMBL2582580 0.82 CTSS (0.48) CTSSCTSKKLK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5747499-A CYCLOPENTAQUINAZOLINE COMPOUNDS CYCLOPENTAQUINAZOLINE COMPOUNDS BRITISH TECHNOLOGY GROUP LIMITED (GB) 1998-05-05 US disclosed
EP-0758328-A1 ANTI-CANCER COMPOUNDS CONTAINING CYCLOPENTAQUINAZOLINE RING BTG INTERNATIONAL LIMITED (GB) 1997-02-19 EP disclosed
WO-1995030673-A1 ANTI-CANCER COMPOUNDS CONTAINING CYCLOPENTAQUINAZOLINE RING BRITISH TECHNOLOGY GROUP LIMITED (GB) 1995-11-16 WO disclosed