SCHEMBL8668207

SCHEMBL8668207

O=C(Nc1c(Cl)cccc1Cl)c1cccc2c1nc(C(F)(F)F)n2CC(=O)N1CCOCC1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 8/20 0.45
PIK3C2B O00750 2/20 0.45
MAPT P10636 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
IL1B P01584 1/20 0.42
P2RX7 Q99572 1/20 0.42
ALDH1A1 P00352 2/20 0.41
GAA P10253 2/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TP53 P04637 1/20 0.41
GRIN1 Q05586 1/20 0.40
GRIN2B Q13224 1/20 0.40
FLT3 P36888 1/20 0.40
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8600301 0.94 PIK3C2B (0.46) IRAK4PIK3C2BMAPTNPC1RAB9A
SCHEMBL8601368 0.89 MAPT (0.46) IRAK4PIK3C2BMAPTALDH1A1GAA
SCHEMBL8598135 0.84 IRAK4 (0.44) IRAK4MAPTNPC1RAB9AGAA
SCHEMBL13990316 0.84 IRAK4 (0.49) IRAK4PIK3C2BMAPTNPC1RAB9A
SCHEMBL8602363 0.84 PIK3C2B (0.52) PIK3C2BMAPTALDH1A1GAASMN1; SMN2
SCHEMBL8598543 0.80 PDE4B (0.43) PIK3C2BP2RX7
SCHEMBL8598985 0.79 PDE4B (0.42) PIK3C2BP2RX7
SCHEMBL8601221 0.79 HPGD (0.46) MAPTALDH1A1HPGDSMN1; SMN2TP53
SCHEMBL8595628 0.79 MAPT (0.52) IRAK4PIK3C2BMAPTALDH1A1GAA
SCHEMBL8596516 0.79 IRAK4 (0.49) IRAK4NPC1RAB9AFLT3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863881-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE IN THE PREVENTION AND/OR THE TREATMENT OF BONE DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-09-16 EP disclosed
WO-1997010219-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE IN THE PREVENTION AND/OR THE TREATMENT OF BONE DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-03-20 WO disclosed